SCHEMBL5363418

SCHEMBL5363418

CC(C)(C)OC(=O)/C=C/c1cc2ccccc2n1Cc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 4/20 0.49
HDAC6 Q9UBN7 2/20 0.42
HDAC10 Q969S8 1/20 0.42
SRC P12931 1/20 0.42
NOD2 Q9HC29 1/20 0.41
NOD1 Q9Y239 1/20 0.41
KMT2A Q03164 1/20 0.40
NR1H2 P55055 3/20 0.40
HPGD P15428 2/20 0.40
KDM4E B2RXH2 2/20 0.40
NR1H3 Q13133 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
HTT P42858 1/20 0.40
LMNA P02545 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5359096 1.00 CCR2 (0.49) CCR2HDAC6HDAC10SRCNOD2
SCHEMBL5427991 0.89 CCR2 (0.43) CCR2HTTMAPTBRD4
SCHEMBL5427985 0.89 CCR2 (0.43) CCR2HTTMAPTBRD4
SCHEMBL5358104 0.85 FDPS (0.40) CCR2KMT2AKDM4EALDH1A1SMN1; SMN2
SCHEMBL5358101 0.85 FDPS (0.40) CCR2KMT2AKDM4EALDH1A1SMN1; SMN2
SCHEMBL5350983 0.85 MAPT (0.43) HDAC6KMT2AKDM4EHDAC1ALDH1A1
SCHEMBL5350992 0.85 MAPT (0.43) HDAC6KMT2AKDM4EHDAC1ALDH1A1
SCHEMBL5369798 0.85 SRD5A2 (0.43) KMT2AKDM4EHDAC8ALDH1A1PPARG
SCHEMBL5372569 0.85 SRD5A2 (0.43) KMT2AKDM4EHDAC8ALDH1A1PPARG
SCHEMBL5362181 0.84 MEN1 (0.42) CCR2KMT2AKDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007134421-A1 2-VINYL INDOLES, PYRIDO AND AZEPINO INDOLE DERIVATIVES, 2-ALKYNYL INDOLES, 2-ALKYNYL BENZO[b]FURANS, THEIR PRECURSORS AND NOVEL PROCESSES FOR THE PREPARATION THEREOF LAUTENS MARK (CA) 2007-11-29 WO disclosed