SCHEMBL5364704

SCHEMBL5364704

Cc1cncc(Cc2ccc(C(=O)O)cc2)c1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 3/20 0.58
HCAR2 Q8TDS4 1/20 0.56
CYP11B1 P15538 10/20 0.51
CYP11B2 P19099 10/20 0.51
CYP3A4 P08684 1/20 0.51
MEN1 O00255 1/20 0.47
LMNA P02545 1/20 0.47
KMT2A Q03164 1/20 0.47
ALDH1A1 P00352 2/20 0.46
RXRA P19793 1/20 0.46
RXRB P28702 1/20 0.46
RXRG P48443 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7431564 0.83 ATM (0.59) CYP11B1CYP11B2CYP3A4ALDH1A1
SCHEMBL21251416 0.81 CYP11B1 (0.57) CYP11B1CYP11B2CYP3A4
SCHEMBL22474091 0.79 CYP11B1 (0.64) CYP11B1CYP11B2CYP3A4
SCHEMBL7877554 0.79 SRD5A2 (0.89) SRD5A2MEN1LMNAKMT2AALDH1A1
Hydrochloric Acid SCHEMBL26136027 0.78 CYP11B1 (0.62) CYP11B1CYP11B2CYP3A4
SCHEMBL68390 0.76 SRD5A2 (0.69) SRD5A2LMNAKMT2AALDH1A1RXRA
SCHEMBL19540958 0.75 CYP11B1 (0.51) CYP11B1CYP11B2CYP3A4
SCHEMBL16880980 0.75 HCAR2 (0.49) SRD5A2HCAR2CYP11B1CYP11B2MEN1
SCHEMBL24088663 0.75 RXRA (0.65) HCAR2ALDH1A1RXRARXRBSMN1; SMN2
SCHEMBL9318665 0.75 MEN1 (0.52) SRD5A2HCAR2CYP11B1CYP11B2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7300934-B2 Benzamide nitriles ROCHE PALO ALTO LLC (US) 2007-11-27 US disclosed
CN-1798729-A Benzamide nitrile derivatives HOFFMANN LA ROCHE (CH) 2006-07-05 CN disclosed
EP-1633701-A1 BENZAMIDE NITRILE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2006-03-15 EP disclosed
WO-2004106285-A1 BENZAMIDE NITRILE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2004-12-09 WO disclosed
US-20040248949-A1 Benzamide nitriles ROCHE PALO ALTO LLC 2004-12-09 US disclosed
WO-2000048993-A1 ARYLAMINOALKYLAMIDES NOVARTIS AG (CH) 2000-08-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040248949-A1 Benzamide nitriles CTSK, CTSS, CMA1 SRD5A2 2667/4885HCAR2 2178/4885CYP11B1 1127/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.