SCHEMBL5366185

SCHEMBL5366185

NC(=O)C1CCN(C(=O)C(N)Cc2ccccc2)CC1

nearest known ligand 0.64

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.64
HDAC8 Q9BY41 3/20 0.59
OPRD1 P41143 1/20 0.59
SMN1; SMN2 Q16637 2/20 0.58
CYP2C19 P33261 1/20 0.58
TACR1 P25103 1/20 0.57
TDP1 Q9NUW8 1/20 0.56
DPP4 P27487 2/20 0.55
FAP Q12884 1/20 0.53
DPP8 Q6V1X1 1/20 0.53
DPP9 Q86TI2 1/20 0.53
DPP7 Q9UHL4 1/20 0.53
ALDH1A1 P00352 1/20 0.53
PLAU P00749 1/20 0.53
PLAUR Q03405 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6583576 1.00 POLB (0.64) POLBHDAC8OPRD1SMN1; SMN2CYP2C19
SCHEMBL5359348 0.86 DPP4 (0.57) POLBDPP4FAPDPP8DPP9
SCHEMBL5367387 0.86 SMN1; SMN2 (0.58) POLBSMN1; SMN2CYP2C19TDP1ALDH1A1
SCHEMBL6161830 0.86 OPRD1 (0.65) POLBHDAC8OPRD1TACR1DPP4
SCHEMBL3133533 0.86 OPRD1 (0.65) POLBHDAC8OPRD1TACR1DPP4
SCHEMBL5374449 0.85 HSD17B10 (0.64) POLBSMN1; SMN2CYP2C19TDP1ALDH1A1
Hydrochloric Acid SCHEMBL6165745 0.84 HDAC8 (0.63) POLBHDAC8OPRD1TACR1DPP4
SCHEMBL7360693 0.84 HPGD (0.66) POLBHDAC8OPRD1TACR1DPP4
Hydrochloric Acid SCHEMBL6163295 0.84 HDAC8 (0.63) POLBHDAC8OPRD1TACR1DPP4
Hydrochloric Acid SCHEMBL6163301 0.84 HDAC8 (0.63) POLBHDAC8OPRD1TACR1DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
CN-1178524-A Di-substituted 1, 4 -piperidine esters and amides having 5-HT4 antagonistic activity BOEHRINGER INGELHEIM ITALIA (IT) 1998-04-08 CN disclosed