SCHEMBL5366189

SCHEMBL5366189

NCC1CCN(C(=O)C(N)Cc2ccccc2)CC1

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 3/20 0.59
OPRD1 P41143 2/20 0.59
OPRK1 P41145 2/20 0.58
DPP4 P27487 3/20 0.55
POLB P06746 1/20 0.55
DPP8 Q6V1X1 2/20 0.53
DPP9 Q86TI2 2/20 0.53
DPP7 Q9UHL4 2/20 0.53
FAP Q12884 1/20 0.53
AKT1 P31749 1/20 0.53
AKT2 P31751 1/20 0.53
AKT3 Q9Y243 1/20 0.53
SMYD3 Q9H7B4 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7361667 0.89 OPRK1 (0.57) HDAC8OPRD1OPRK1DPP4POLB
SCHEMBL2375481 0.89 OPRK1 (0.71) HDAC8OPRD1OPRK1DPP4POLB
SCHEMBL2375476 0.89 OPRK1 (0.71) HDAC8OPRD1OPRK1DPP4POLB
SCHEMBL5359350 0.86 DPP4 (0.57) DPP4DPP8DPP9DPP7FAP
SCHEMBL5367391 0.86 CHRM1 (0.48) OPRD1OPRK1POLB
SCHEMBL3133533 0.86 OPRD1 (0.65) HDAC8OPRD1OPRK1DPP4POLB
SCHEMBL6161830 0.86 OPRD1 (0.65) HDAC8OPRD1OPRK1DPP4POLB
SCHEMBL2375638 0.85 OPRD1 (0.61) HDAC8OPRD1OPRK1DPP4POLB
SCHEMBL7364618 0.85 OPRK1 (0.57) HDAC8OPRD1OPRK1DPP4POLB
SCHEMBL2375634 0.85 OPRD1 (0.61) HDAC8OPRD1OPRK1DPP4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed