SCHEMBL5366982

SCHEMBL5366982

Cc1ccc(CN2CCC(CNC(=O)c3ccc(O)cc3)C(O)C2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 2/20 0.53
KCNH2 Q12809 1/20 0.53
CACNA1I Q9P0X4 1/20 0.53
GAA P10253 3/20 0.48
CHRM4 P08173 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.47
UBE2N P61088 1/20 0.46
TP53 P04637 2/20 0.45
HDAC3 O15379 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC10 Q969S8 1/20 0.45
HDAC11 Q96DB2 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
HDAC9 Q9UKV0 1/20 0.45
HDAC5 Q9UQL6 1/20 0.45
LMNA P02545 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14425271 1.00 CCR2 (0.53) CCR2KCNH2CACNA1IGAACHRM4
SCHEMBL5359305 0.83 KCNH2 (0.73) CCR2KCNH2CACNA1IGAACHRM4
SCHEMBL14425272 0.82 LMNA (0.45) CCR2GAACHRM4TP53HDAC3
SCHEMBL5374660 0.82 LMNA (0.45) CCR2GAACHRM4TP53HDAC3
SCHEMBL14425270 0.77 CHRM4 (0.53) KCNH2CHRM4HDAC3HDAC4HDAC1
SCHEMBL5368709 0.77 CHRM4 (0.53) KCNH2CHRM4HDAC3HDAC4HDAC1
SCHEMBL5378277 0.74 HDAC3 (0.71) CHRM4HDAC3HDAC4HDAC1HDAC7
SCHEMBL5368040 0.73 CCR2 (0.69) CCR2KCNH2CACNA1ICHRM4HDAC3
SCHEMBL5368811 0.72 HDAC3 (0.64) CCR2KCNH2CACNA1IGAACHRM4
SCHEMBL5365422 0.72 TPSAB1 (0.63) KCNH2CACNA1ILMNAKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed