SCHEMBL5368709

SCHEMBL5368709

O=C(NCC1CCN(CCCc2ccccc2)CC1O)c1ccc(O)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 2/20 0.53
CHRNB2 P17787 1/20 0.48
CHRNA4 P43681 1/20 0.48
DRD4 P21917 1/20 0.47
HDAC3 O15379 2/20 0.46
HDAC4 P56524 2/20 0.46
HDAC1 Q13547 2/20 0.46
HDAC7 Q8WUI4 2/20 0.46
HDAC2 Q92769 2/20 0.46
HDAC10 Q969S8 2/20 0.46
HDAC11 Q96DB2 2/20 0.46
HDAC8 Q9BY41 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
HDAC9 Q9UKV0 2/20 0.46
HDAC5 Q9UQL6 2/20 0.46
KCNH2 Q12809 1/20 0.46
LTA4H P09960 1/20 0.46
SLC6A2 P23975 1/20 0.45
SLC6A4 P31645 1/20 0.45
CCR3 P51677 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14425270 1.00 CHRM4 (0.53) CHRM4CHRNB2CHRNA4DRD4HDAC3
SCHEMBL5370678 0.84 CHRM4 (0.63) CHRM4HDAC3HDAC4HDAC1HDAC7
SCHEMBL5375113 0.82 CHRNB2 (0.69) CHRM4CHRNB2CHRNA4LTA4HSLC6A2
SCHEMBL5365173 0.80 ADRB1 (0.54) CHRM4CHRNB2CHRNA4DRD4HDAC4
SCHEMBL5368664 0.80 DRD4 (0.54) CHRM4CHRNB2CHRNA4DRD4
SCHEMBL14425262 0.78 F2 (0.53) HDAC1HDAC6
SCHEMBL5371368 0.78 F2 (0.53) HDAC1HDAC6
SCHEMBL14425224 0.78 F2 (0.53) HDAC1HDAC6
SCHEMBL14425190 0.78 F2 (0.53) HDAC1HDAC6
SCHEMBL5366982 0.77 CCR2 (0.53) CHRM4DRD4HDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed