SCHEMBL5368683

SCHEMBL5368683

Cc1cc(Cc2ccc(Cl)c(Oc3cccc4[nH]ccc34)c2F)n[nH]c1=O

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
RHEB Q15382 7/20 0.43
SLC5A2 P31639 1/20 0.39
TRPA1 O75762 1/20 0.38
SCN9A Q15858 1/20 0.36
P2RX7 Q99572 1/20 0.34
DAO P14920 2/20 0.33
NR3C1 P04150 1/20 0.32
LMNA P02545 1/20 0.31
HTT P42858 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
MEN1 O00255 1/20 0.31
MAPT P10636 1/20 0.31
MAPK1 P28482 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14570780 0.89 CYP3A4 (0.44) CYP3A4CYP2C9CYP2C19RHEBSLC5A2
SCHEMBL4268874 0.86 CYP3A4 (0.56) CYP3A4CYP2C9CYP2C19SLC5A2P2RX7
SCHEMBL5364861 0.85 RHEB (0.44) CYP3A4CYP2C9CYP2C19RHEBTRPA1
SCHEMBL5364607 0.83 CYP3A4 (0.56) CYP3A4CYP2C9CYP2C19SLC5A2SCN9A
SCHEMBL5373905 0.80 CYP3A4 (0.56) CYP3A4CYP2C9CYP2C19SLC5A2P2RX7
SCHEMBL5368877 0.80 CYP3A4 (0.70) CYP3A4CYP2C9CYP2C19RHEBSLC5A2
SCHEMBL5209110 0.79 CYP3A4 (0.59) CYP3A4CYP2C9CYP2C19SLC5A2DAO
SCHEMBL5373748 0.78 CYP3A4 (0.56) CYP3A4CYP2C9CYP2C19SLC5A2DAO
SCHEMBL5370974 0.78 CYP3A4 (0.73) CYP3A4CYP2C9CYP2C19SLC5A2P2RX7
SCHEMBL5374165 0.77 CYP3A4 (0.74) CYP3A4CYP2C9CYP2C19SLC5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed