SCHEMBL5364607

SCHEMBL5364607

Cc1cc(Cc2ccc(Cl)c(Oc3cccc4ncccc34)c2F)n[nH]c1=O

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
SLC5A2 P31639 1/20 0.38
SCN9A Q15858 1/20 0.37
NR3C1 P04150 4/20 0.36
PARP1 P09874 2/20 0.35
P2RX7 Q99572 1/20 0.35
NPBWR1 P48145 1/20 0.35
DAO P14920 2/20 0.34
DRD1 P21728 1/20 0.34
PDE10A Q9Y233 2/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
SYK P43405 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5373905 0.87 CYP3A4 (0.56) CYP3A4CYP2C9CYP2C19SLC5A2PARP1
SCHEMBL5368683 0.83 CYP3A4 (0.56) CYP3A4CYP2C9CYP2C19SLC5A2SCN9A
SCHEMBL4268874 0.80 CYP3A4 (0.56) CYP3A4CYP2C9CYP2C19SLC5A2P2RX7
SCHEMBL5373748 0.79 CYP3A4 (0.56) CYP3A4CYP2C9CYP2C19SLC5A2DAO
SCHEMBL5368877 0.79 CYP3A4 (0.70) CYP3A4CYP2C9CYP2C19SLC5A2NPBWR1
SCHEMBL5370974 0.77 CYP3A4 (0.73) CYP3A4CYP2C9CYP2C19SLC5A2PARP1
SCHEMBL5209110 0.76 CYP3A4 (0.59) CYP3A4CYP2C9CYP2C19SLC5A2DAO
SCHEMBL5374165 0.76 CYP3A4 (0.74) CYP3A4CYP2C9CYP2C19SLC5A2DRD1
SCHEMBL5368624 0.75 CYP3A4 (0.80) CYP3A4CYP2C9CYP2C19SLC5A2NPBWR1
SCHEMBL4274657 0.73 CYP3A4 (0.91) CYP3A4CYP2C9CYP2C19SLC5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed