SCHEMBL5373748

SCHEMBL5373748

Cc1cc(Cc2ccc(Cl)c(Oc3cccc4ccc[n+]([O-])c34)c2F)n[nH]c1=O

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.56
CYP2C9 P11712 3/20 0.56
CYP2C19 P33261 3/20 0.56
SLC5A2 P31639 1/20 0.37
DAO P14920 6/20 0.35
LMNA P02545 1/20 0.32
HTT P42858 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CYP1A2 P05177 2/20 0.30
PTGER1 P34995 2/20 0.30
ADORA2A P29274 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5373905 0.82 CYP3A4 (0.56) CYP3A4CYP2C9CYP2C19SLC5A2DAO
SCHEMBL4268874 0.82 CYP3A4 (0.56) CYP3A4CYP2C9CYP2C19SLC5A2DAO
SCHEMBL5368877 0.80 CYP3A4 (0.70) CYP3A4CYP2C9CYP2C19SLC5A2DAO
SCHEMBL5364607 0.79 CYP3A4 (0.56) CYP3A4CYP2C9CYP2C19SLC5A2DAO
SCHEMBL5368683 0.78 CYP3A4 (0.56) CYP3A4CYP2C9CYP2C19SLC5A2DAO
SCHEMBL5370974 0.78 CYP3A4 (0.73) CYP3A4CYP2C9CYP2C19SLC5A2DAO
SCHEMBL5368624 0.76 CYP3A4 (0.80) CYP3A4CYP2C9CYP2C19SLC5A2
SCHEMBL4278760 0.76 CYP3A4 (0.62) CYP3A4CYP2C9CYP2C19SLC5A2
SCHEMBL5374165 0.75 CYP3A4 (0.74) CYP3A4CYP2C9CYP2C19SLC5A2
SCHEMBL5209110 0.75 CYP3A4 (0.59) CYP3A4CYP2C9CYP2C19SLC5A2DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed