SCHEMBL538290

SCHEMBL538290

CN(C)C(=O)c1ccccc1N

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.55
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
KDM4E B2RXH2 6/20 0.55
ALDH1A1 P00352 12/20 0.53
HSD17B10 Q99714 6/20 0.53
CFTR P13569 1/20 0.53
MAPT P10636 4/20 0.50
GAA P10253 2/20 0.50
KEAP1 Q14145 1/20 0.49
HPGD P15428 4/20 0.44
SLC6A4 P31645 1/20 0.43
TP53 P04637 2/20 0.42
TSHR P16473 2/20 0.42
POLB P06746 1/20 0.41
MMP2 P08253 1/20 0.41
ALOX15 P16050 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30598338 1.00 SMN1; SMN2 (0.55) SMN1; SMN2MEN1KMT2AKDM4EALDH1A1
Hydrochloric Acid SCHEMBL15569994 0.98 SMN1; SMN2 (0.53) SMN1; SMN2MEN1KMT2AKDM4EALDH1A1
SCHEMBL9254635 0.85 KDM4E (0.53) SMN1; SMN2MEN1KMT2AKDM4EALDH1A1
SCHEMBL28248149 0.84 KMT2A (0.51) SMN1; SMN2MEN1KMT2AKDM4EALDH1A1
SCHEMBL188296 0.84 MEN1 (0.65) SMN1; SMN2MEN1KMT2AKDM4EALDH1A1
SCHEMBL27938205 0.83 KDM4E (0.51) SMN1; SMN2MEN1KMT2AKDM4EALDH1A1
SCHEMBL8082335 0.83 MEN1 (0.47) SMN1; SMN2MEN1KMT2AKDM4EALDH1A1
SCHEMBL13254933 0.82 CYP3A4 (0.48) SMN1; SMN2MEN1KMT2AKDM4EALDH1A1
SCHEMBL1706450 0.82 MMP2 (0.60) SMN1; SMN2MEN1KMT2AALDH1A1HSD17B10
SCHEMBL25078318 0.80 MEN1 (0.44) SMN1; SMN2MEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 156 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101250135-A Synthetic method of 2-amino-N, N-dimethylbenzamide YANCHENG LVYE CHEMICAL INDUSTR (CN) 2008-08-27 CN claimed
US-12612424-B2 HPK1 inhibitors and uses thereof REGOR PHARMACEUTICALS, INC. (US) 2026-04-28 US disclosed
CN-114555585-B HPK1 inhibitors and uses thereof 锐格药业公司 2025-02-11 CN disclosed
US-20220389037-A1 HPK1 INHIBITORS AND USES THEREOF REGOR PHARMACEUTICALS, INC. 2022-12-08 US disclosed
WO-2022214008-A1 HIGHLY ACTIVE HPK1 KINASE INHIBITOR 杭州阿诺生物医药科技有限公司 2022-10-13 WO disclosed
CN-114555585-A HPK1 inhibitors and uses thereof 上海齐鲁锐格医药研发有限公司 2022-05-27 CN disclosed
EP-3994133-A1 HPK1 INHIBITORS AND USES THEREOF Qilu Regor Therapeutics Inc. (CN) 2022-05-11 EP disclosed
US-10752624-B2 Kinase inhibitors ORIGENIS GMBH (DE) 2020-08-25 US disclosed
EP-3325475-B1 OXADIAZOLE DERIVATIVES USEFUL AS HDAC INHIBITORS TAKEDA PHARMACEUTICALS CO (JP) 2020-03-18 EP disclosed
US-10308643-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2019-06-04 US disclosed
WO-1998040361-A1 AMINOSULFONYLUREAS WITH HERBICIDAL ACTIVITY ISAGRO RICERCA S.R.L. (IT) 1998-09-17 WO disclosed
US-5688795-A URINARY TRACTS OBSTRUCTION SYNTEX (U.S.A.) INC. (US) 1997-11-18 US disclosed
EP-0711757-A1 3-(4-phenylpiperazin-1-yl)propyl-amino, thio and oxy -pyridine, pyrimidine and benzene derivatives as alpha1-adrenoceptor antagonists F. Hoffmann-La Roche AG (CH) 1996-05-15 EP disclosed
EP-0317859-B1 AZO DYES CONTAINING POLYETHYLENIMINE BASF Aktiengesellschaft (DE) 1991-11-27 EP disclosed
US-4962190-A PRINTING, DYEING CELLULOSE CONTAINING MATERIAL BASF AKTIENGESELLSCHAFT (DE) 1990-10-09 US disclosed
US-4835312-A Production process of N-substituted amide compounds MITSUI CHEMICALS, INCORPORATED (JP) 1989-05-30 US disclosed
EP-0084853-B1 PROCESS FOR THE PREPARATION OF 1,8-NAPHTHOLACTAM COMPOUNDS CIBA-GEIGY AG (CH) 1986-11-12 EP disclosed
US-4515963-A AMIDATIUON OF NAPHTHOLACTONE CIBA GEIGY AG (CH) 1985-05-07 US disclosed
EP-0084853-A1 Process for the preparation of 1,8-naphtholactam compounds CIBA-GEIGY AG (CH) 1983-08-03 EP disclosed
US-4163059-A Pesticidally active 4,5-dichloro-3-substituted-phenylimino-1,2-dithiolenes BAYER AKTIENGESELLSCHAFT (DE) 1979-07-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12612424-B2 HPK1 inhibitors and uses thereof NEK11, NEK1, CSNK1A1 SMN1; SMN2 3906/4885MEN1 3442/4885KMT2A 1353/4885
US-20220389037-A1 HPK1 INHIBITORS AND USES THEREOF HIPK1, SIK1, PGK1 SMN1; SMN2 3998/4885MEN1 1442/4885KMT2A 2256/4885
US-10308643-B2 Heterocyclic compound HDAC1, HDAC11, HDAC5 SMN1; SMN2 38/4885MEN1 2720/4885KMT2A 47/4885
US-10752624-B2 Kinase inhibitors LRRK2, MYLK2, MYLK SMN1; SMN2 986/4885MEN1 636/4885KMT2A 929/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.