SCHEMBL5402346

SCHEMBL5402346

O=c1[nH]c(=O)n(Cc2ccccc2)c(=O)n1O

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.50
ALDH1A1 P00352 3/20 0.50
ERCC5 P28715 2/20 0.50
FEN1 P39748 2/20 0.50
KDM4E B2RXH2 2/20 0.50
CYP3A4 P08684 2/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
ERCC1 P07992 1/20 0.50
ERCC4 Q92889 1/20 0.50
PARN O95453 1/20 0.48
CNOT7 Q9UIV1 1/20 0.48
GSK3A P49840 2/20 0.47
GSK3B P49841 2/20 0.47
DAO P14920 2/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
PNP P00491 1/20 0.44
LMNA P02545 1/20 0.44
HTT P42858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL38658744 0.79 KMT2A (0.56) HPGDALDH1A1KDM4ECYP3A4SMN1; SMN2
SCHEMBL14950255 0.77 MAPK8 (0.56) HPGDALDH1A1KDM4ECYP3A4SMN1; SMN2
SCHEMBL8985073 0.76 GSK3B (0.67) HPGDALDH1A1KDM4ECYP3A4SMN1; SMN2
SCHEMBL2337883 0.75 HPGD (0.58) HPGDALDH1A1KDM4ECYP3A4SMN1; SMN2
SCHEMBL11679530 0.74 HPGD (0.45) HPGDALDH1A1KDM4ECYP3A4SMN1; SMN2
SCHEMBL28160033 0.73 HPGD (0.51) HPGDALDH1A1KDM4ECYP3A4SMN1; SMN2
SCHEMBL9453672 0.72 GSK3A (0.57) HPGDALDH1A1KDM4ECYP3A4SMN1; SMN2
SCHEMBL19783871 0.71 GSK3B (0.51) HPGDALDH1A1KDM4ECYP3A4SMN1; SMN2
SCHEMBL10859990 0.71 LGMN (0.66) HPGDALDH1A1KDM4ECYP3A4SMN1; SMN2
SCHEMBL10070157 0.71 PGR (0.66) ALDH1A1ERCC5FEN1KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5624982-A BENZOTRIAZOLE COMPOUNDS FOR LIGHT STABILIZERS OF TETRAMETHYL PIPERIDINYL SEBACATE FOR STYRENE POLYMERS BAYER ANTWERPEN SA/NV (BE) 1997-04-29 US claimed
EP-0736064-A1 STABILIZER SYSTEM FOR NON YELLOWING POLYMER COMPOSITION BAYER ANTWERPEN N.V. (BE) 1996-10-09 EP claimed
WO-1995015358-A1 STABILIZER SYSTEM FOR NON YELLOWING POLYMER COMPOSITION BAYER ANTWERPEN SA/NV (BE) 1995-06-08 WO claimed
US-7259198-B2 Ultraviolet radiation stabilized polyolefins EXXONMOBIL CHEMICAL PATENTS INC. (US) 2007-08-21 US disclosed
US-5624982-A BENZOTRIAZOLE COMPOUNDS FOR LIGHT STABILIZERS OF TETRAMETHYL PIPERIDINYL SEBACATE FOR STYRENE POLYMERS BAYER ANTWERPEN SA/NV (BE) 1997-04-29 US disclosed
EP-0736064-A1 STABILIZER SYSTEM FOR NON YELLOWING POLYMER COMPOSITION BAYER ANTWERPEN N.V. (BE) 1996-10-09 EP disclosed
US-5492948-A STABILIZER FOR STYRENE POLYMERS CONSISTING OF A BENZOTRIAZOLE, OLIGOMERIC CONDENSATE OF 2,4-DICHLORO-6-MORPHOLINO-S-TRIAZINE AND N,N*-/2,2,6,6-TETRAMETHYLPIPERIDYL/HEXAMETHYLENEDIAMINE, TRIS/3,5-DI-TERT-BUTYL-4-HYDROXYBENZYL/ ISOCYANURATE MONSANTO COMPANY (US) 1996-02-20 US disclosed
WO-1995015358-A1 STABILIZER SYSTEM FOR NON YELLOWING POLYMER COMPOSITION BAYER ANTWERPEN SA/NV (BE) 1995-06-08 WO disclosed