SCHEMBL5404643

SCHEMBL5404643

O=[N+]([O-])c1[c]cccc1-c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
EIF4E P06730 2/20 0.38
CYP3A4 P08684 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
HIF1A Q16665 1/20 0.38
TXNRD1 Q16881 1/20 0.38
TXNRD3 Q86VQ6 1/20 0.38
TXNRD2 Q9NNW7 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
P2RX1 P51575 2/20 0.36
MASP2 O00187 1/20 0.35
F2 P00734 1/20 0.35
KIF11 P52732 1/20 0.34
LMNA P02545 2/20 0.33
PARP1 P09874 1/20 0.33
FBP1 P09467 1/20 0.33
PTPN5 P54829 1/20 0.33
SCN2A Q99250 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6191439 0.80 EIF4E (0.35) ALDH1A1EIF4ECYP3A4HIF1ATDP1
SCHEMBL6232168 0.77 ALDH1A1 (0.36) ALDH1A1CYP3A4TSHRHIF1ATDP1
SCHEMBL3535919 0.76 ALDH1A1 (0.53) ALDH1A1CYP3A4HPGDHIF1ATDP1
SCHEMBL15868446 0.75 ALDH1A1 (0.58) ALDH1A1EIF4ECYP3A4HPGDALOX15
SCHEMBL6194171 0.75 PTGS2 (0.40) ALDH1A1EIF4ETDP1FBP1MAPT
SCHEMBL6192872 0.75 FBP1 (0.40) ALDH1A1EIF4ETDP1FBP1MAPT
SCHEMBL6683239 0.73 HTR7 (0.42) ALDH1A1CYP3A4TDP1LMNASCN2A
SCHEMBL5150349 0.73 TSHR (0.48) ALDH1A1ALOX15TSHRTDP1LMNA
SCHEMBL3556690 0.73 ALDH1A1 (0.34) ALDH1A1CYP3A4HPGDALOX15TSHR
SCHEMBL6191701 0.72 PTGS2 (0.40) ALDH1A1EIF4EHPGDTSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007518825-A 2007-07-12 JP claimed
EP-1706399-A1 POLYETHYLENE GLYCOL CONJUGATES OF HETEROCYCLOALKYL CARBOXAMIDO PROPANOIC ACIDS Elan Pharmaceuticals, Inc. (US) 2006-10-04 EP claimed
WO-2005070921-A1 POLYETHYLENE GLYCOL CONJUGATES OF HETEROCYCLOALKYL CARBOXAMIDO PROPANOIC ACIDS ELAN PHARMACEUTICALS, INC. (US) 2005-08-04 WO claimed