SCHEMBL5405855

SCHEMBL5405855

COc1ccc2c(c(C=O)cn2C)c1N

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.46
IMPDH2 P12268 1/20 0.41
KDM4E B2RXH2 2/20 0.41
ERN1 O75460 5/20 0.36
HTR1D P28221 1/20 0.36
HTR1B P28222 1/20 0.36
TDP1 Q9NUW8 2/20 0.36
TSHR P16473 2/20 0.36
KDR P35968 1/20 0.35
NPC1 O15118 1/20 0.35
MAPT P10636 1/20 0.35
RAB9A P51151 1/20 0.35
TLR2 O60603 1/20 0.35
TLR1 Q15399 1/20 0.35
TLR6 Q9Y2C9 1/20 0.35
NQO2 P16083 1/20 0.34
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3690189 0.78 NQO2 (0.53) ALDH1A1IMPDH2KDM4EERN1HTR1D
SCHEMBL1093104 0.78 ALDH1A1 (0.51) ALDH1A1IMPDH2KDM4EERN1TDP1
SCHEMBL19865517 0.73 NQO2 (0.42) ALDH1A1KDM4EMAPTRAB9ANQO2
SCHEMBL31205479 0.73 ALDH1A1 (0.46) ALDH1A1IMPDH2KDM4EERN1HTR1D
SCHEMBL8818184 0.72 ALDH1A1 (0.41) ALDH1A1KDM4EERN1TSHRNPC1
SCHEMBL30045931 0.72 ALDH1A1 (0.41) ALDH1A1KDM4EERN1TSHRNPC1
SCHEMBL1451216 0.71 ALDH1A1 (0.57) ALDH1A1IMPDH2KDM4EERN1TDP1
SCHEMBL27756846 0.68 ALDH1A1 (0.47) ALDH1A1KDM4EERN1TDP1TSHR
SCHEMBL1138275 0.67 PTGER3 (0.55) ALDH1A1IMPDH2
SCHEMBL1043732 0.66 ERN1 (0.61) ALDH1A1KDM4EERN1TDP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018031662-A1 PYRROLOBENZODIAZEPINE PRODRUGS AND ANTIBODY CONJUGATES THEREOF GENENTECH, INC. (US) 2018-02-15 WO disclosed
US-7304046-B2 Phosphoramide compounds PURDUE RESEARCH FOUNDATION (US) 2007-12-04 US disclosed
US-7304046-B2 Phosphoramide compounds PURDUE RESEARCH FOUNDATION (US) 2007-12-04 US disclosed
US-7304046-B2 Phosphoramide compounds PURDUE RESEARCH FOUNDATION (US) 2007-12-04 US disclosed
US-20040176332-A1 Phosphoramide compounds PURDUE RESEARCH FOUNDATION 2004-09-09 US disclosed
US-6656926-B2 For therapy and prophylaxis of cancer PURDUE RESEARCH FOUNDATION 2003-12-02 US disclosed
US-20030008850-A1 For therapy and prophylaxis of cancer NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2003-01-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040176332-A1 Phosphoramide compounds RB1, RRM2B, RRM1 ALDH1A1 1067/4885IMPDH2 892/4885KDM4E 3140/4885
US-20030008850-A1 For therapy and prophylaxis of cancer BRCA1, RRM2B, FOLR1 ALDH1A1 27/4885IMPDH2 1436/4885KDM4E 3105/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.