SCHEMBL5408629

SCHEMBL5408629

COc1ccc(-c2ccc(C#N)cc2)nc1C=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 1/20 0.43
CYP1B1 Q16678 1/20 0.43
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
KDM4E B2RXH2 3/20 0.40
ALDH1A1 P00352 3/20 0.40
F2RL3 Q96RI0 1/20 0.40
GAA P10253 2/20 0.40
MCHR1 Q99705 1/20 0.39
ACLY P53396 1/20 0.38
MAPT P10636 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
GLA P06280 1/20 0.37
GFER P55789 1/20 0.37
GRM2 Q14416 1/20 0.37
FGFR4 P22455 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4799749 0.80 TDO2 (0.51) MEN1KMT2AKDM4EALDH1A1GAA
SCHEMBL15577522 0.79 KDM4E (0.55) CYP1A1CYP1B1MEN1KMT2AKDM4E
SCHEMBL18532398 0.79 MAOB (0.43) CYP1A1CYP1B1MEN1KMT2AF2RL3
SCHEMBL14435490 0.74 SCN9A (0.39) MEN1KMT2AKDM4EGAAMAPT
SCHEMBL15577732 0.73 ALDH1A1 (0.46) CYP1A1CYP1B1MEN1KMT2AKDM4E
SCHEMBL4600422 0.72 ERN1 (0.50) MEN1KMT2AKDM4EALDH1A1ACLY
SCHEMBL12539439 0.71 TRPV3 (0.53) KMT2AHPGDHSD17B10
SCHEMBL6061082 0.70 HPGD (0.47) KDM4EALDH1A1L3MBTL1KITHPGD
SCHEMBL24137877 0.70 KDM1A (0.39) KDM4EALDH1A1MCHR1CYP2C9CYP2C19
SCHEMBL8433481 0.70 ALDH1A1 (0.51) ALDH1A1ACLYKITHPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007089031-A1 PIPERIDINE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-08-09 WO disclosed