SCHEMBL5408973

SCHEMBL5408973

Cc1ccc(CCN(CCC(=O)O)C(=O)c2ccccc2-c2ccccc2C(=O)NCc2ccc(C(C)(C)C)cc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 8/20 0.52
EPHX2 P34913 7/20 0.52
ALDH1A1 P00352 4/20 0.48
LMNA P02545 1/20 0.46
RAB9A P51151 1/20 0.46
KDM4E B2RXH2 2/20 0.44
HPGD P15428 2/20 0.44
ESRRG P62508 2/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
CHRNB2 P17787 1/20 0.41
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41
CHRNA4 P43681 1/20 0.41
PPARA Q07869 2/20 0.41
PPARG P37231 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5402883 0.95 NR1H4 (0.55) NR1H4EPHX2ALDH1A1LMNARAB9A
SCHEMBL5402458 0.93 ALDH1A1 (0.55) ALDH1A1LMNAKDM4EHPGDHDAC1
SCHEMBL5418399 0.92 ALDH1A1 (0.57) ALDH1A1LMNARAB9AKDM4EHPGD
SCHEMBL5399793 0.92 ALDH1A1 (0.57) ALDH1A1LMNARAB9AKDM4EHPGD
SCHEMBL5416724 0.91 NR1H4 (0.50) NR1H4EPHX2ALDH1A1LMNARAB9A
SCHEMBL5405971 0.90 NR1H4 (0.54) NR1H4EPHX2ALDH1A1LMNARAB9A
SCHEMBL5405685 0.90 EPHX2 (0.53) NR1H4EPHX2ALDH1A1LMNARAB9A
SCHEMBL5402812 0.89 NR1H4 (0.47) NR1H4EPHX2ALDH1A1LMNARAB9A
SCHEMBL5402442 0.89 ALDH1A1 (0.50) ALDH1A1LMNARAB9AKDM4EHPGD
SCHEMBL5399508 0.89 ALDH1A1 (0.50) ALDH1A1LMNAKDM4EHPGDHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7285680-B2 β-alanine derivatives and the use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2007-10-23 US disclosed
US-20050256160-A1 Beta-alanine derivatives and the use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2005-11-17 US disclosed
EP-1533294-A1 BETA-ALANINE DERIVATIVE AND USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2005-05-25 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050256160-A1 Beta-alanine derivatives and the use thereof TGFB1, PML, APOB NR1H4 546/4885EPHX2 2105/4885ALDH1A1 1256/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.