SCHEMBL5402883

SCHEMBL5402883

CC(C)(C)c1ccc(CNC(=O)c2ccccc2-c2ccccc2C(=O)N(CCC(=O)O)CCc2ccccc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 9/20 0.55
EPHX2 P34913 8/20 0.55
RAB9A P51151 2/20 0.51
LMNA P02545 1/20 0.51
CHRNB2 P17787 1/20 0.46
CHRNB4 P30926 1/20 0.46
CHRNA3 P32297 1/20 0.46
CHRNA4 P43681 1/20 0.46
ESRRG P62508 2/20 0.46
NPC1 O15118 1/20 0.44
PPARG P37231 1/20 0.43
ALDH1A1 P00352 1/20 0.43
EGFR P00533 1/20 0.42
HDAC3 O15379 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
MAOA P21397 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5408973 0.95 NR1H4 (0.52) NR1H4EPHX2RAB9ALMNACHRNB2
SCHEMBL5405971 0.95 NR1H4 (0.54) NR1H4EPHX2RAB9ALMNACHRNB2
SCHEMBL5416724 0.93 NR1H4 (0.50) NR1H4EPHX2RAB9ALMNACHRNB2
SCHEMBL5405685 0.93 EPHX2 (0.53) NR1H4EPHX2RAB9ALMNANPC1
SCHEMBL5405681 0.91 ALDH1A1 (0.52) NR1H4EPHX2RAB9ALMNANPC1
SCHEMBL5392424 0.91 CA2 (0.54) NR1H4EPHX2ALDH1A1
SCHEMBL5397527 0.91 NR1H4 (0.54) NR1H4EPHX2RAB9ALMNAESRRG
SCHEMBL5409367 0.91 LMNA (0.52) NR1H4EPHX2RAB9ALMNACHRNB2
SCHEMBL5409780 0.91 CHRNB2 (0.56) RAB9ALMNACHRNB2CHRNB4CHRNA3
SCHEMBL5402812 0.90 NR1H4 (0.47) NR1H4EPHX2RAB9ALMNACHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7285680-B2 β-alanine derivatives and the use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2007-10-23 US disclosed
US-20050256160-A1 Beta-alanine derivatives and the use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2005-11-17 US disclosed
EP-1533294-A1 BETA-ALANINE DERIVATIVE AND USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2005-05-25 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050256160-A1 Beta-alanine derivatives and the use thereof TGFB1, PML, APOB NR1H4 546/4885EPHX2 2105/4885RAB9A 3132/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.