SCHEMBL542952

SCHEMBL542952

O=C(OCc1cc(C(F)(F)F)ccc1F)N1CCCCC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.49
HPGD P15428 3/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
TSHR P16473 1/20 0.46
LMNA P02545 2/20 0.45
POLB P06746 1/20 0.45
MGLL Q99685 2/20 0.44
ABHD6 Q9BV23 2/20 0.44
PLA2G7 Q13093 1/20 0.44
ENPP2 Q13822 3/20 0.43
ATXN2 Q99700 3/20 0.43
CA2 P00918 1/20 0.43
CYP2D6 P10635 1/20 0.43
LIPE Q05469 2/20 0.42
BCHE P06276 1/20 0.42
ALDH1A1 P00352 1/20 0.42
RAB9A P51151 2/20 0.41
MAPK1 P28482 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL543019 0.90 ENPP2 (0.52) IDO1HPGDMEN1KMT2ATSHR
SCHEMBL543231 0.80 MEN1 (0.55) HPGDMEN1KMT2ATSHRENPP2
SCHEMBL542677 0.78 MEN1 (0.53) HPGDMEN1KMT2ATSHRENPP2
SCHEMBL16825194 0.78 GRIN2B (0.57) MEN1KMT2ATSHRLMNAPOLB
SCHEMBL28032629 0.78 KMT2A (0.64) IDO1HPGDMEN1KMT2ALMNA
SCHEMBL4682405 0.78 ENPP2 (0.52) IDO1HPGDLMNAENPP2ATXN2
SCHEMBL6236300 0.78 ENPP2 (0.50) IDO1MEN1KMT2AMGLLABHD6
SCHEMBL543132 0.77 TACR1 (0.49) IDO1HPGDMEN1KMT2ATSHR
Hydrochloric Acid SCHEMBL4682398 0.77 ENPP2 (0.51) IDO1HPGDLMNAENPP2ATXN2
SCHEMBL14255640 0.76 IDO1 (0.58) IDO1HPGDPOLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414330-A2 PIPERIDINE AND PIPERAZINE DERIVATIVES AS AUTOTAXIN INHIBITORS Merck Patent GmbH (DE) 2012-02-08 EP claimed
WO-2010115491-A2 PIPERIDINE AND PIPERAZINE DERIVATIVES AS AUTOTAXIN INHIBITORS MERCK PATENT GMBH (DE) 2010-10-14 WO claimed