SCHEMBL6236300

SCHEMBL6236300

O=C(OCc1ccc(C(F)(F)F)cc1F)N1CCOCC1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 3/20 0.50
ATXN2 Q99700 3/20 0.50
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
MGLL Q99685 1/20 0.48
ABHD6 Q9BV23 1/20 0.48
IDO1 P14902 1/20 0.47
AKR1C3 P42330 1/20 0.45
FKBP1A P62942 1/20 0.45
GAA P10253 1/20 0.44
EPHX2 P34913 2/20 0.44
LIPE Q05469 1/20 0.44
ALOX5AP P20292 2/20 0.43
FEN1 P39748 2/20 0.43
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL543019 0.88 ENPP2 (0.52) ENPP2ATXN2MEN1KMT2AMGLL
SCHEMBL4682405 0.85 ENPP2 (0.52) ENPP2ATXN2IDO1RAB9A
SCHEMBL6235265 0.85 MEN1 (0.53) MEN1KMT2ANPSR1IDO1FKBP1A
Hydrochloric Acid SCHEMBL4682398 0.84 ENPP2 (0.51) ENPP2ATXN2IDO1RAB9A
SCHEMBL542952 0.78 IDO1 (0.49) ENPP2ATXN2MEN1KMT2AMGLL
SCHEMBL14425370 0.76 ENPP2 (0.42) ENPP2ATXN2MEN1KMT2A
SCHEMBL5360981 0.76 ENPP2 (0.42) ENPP2ATXN2MEN1KMT2A
SCHEMBL6235843 0.76 MEN1 (0.55) ENPP2ATXN2MEN1KMT2ANPSR1
SCHEMBL14255637 0.74 IDO1 (0.58) ENPP2ATXN2IDO1GAA
SCHEMBL6235042 0.73 MEN1 (0.62) ENPP2ATXN2MEN1KMT2ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1390034-A4 N-SUBSTITUTED NONARYL-HETEROCYCLO AMIDYL NMDA/NR2B ANTAGONISTS MERCK & CO INC (US) 2005-07-13 EP disclosed
EP-1390034-A1 N-SUBSTITUTED NONARYL-HETEROCYCLO AMIDYL NMDA/NR2B ANTAGONISTS Merck & Co., Inc. (US) 2004-02-25 EP disclosed
WO-2002080928-A1 N-SUBSTITUTED NONARYL-HETEROCYCLO AMIDYL NMDA/NR2B ANTAGONISTS MERCK & CO., INC. (US) 2002-10-17 WO disclosed