SCHEMBL5434147

SCHEMBL5434147

COC(=O)c1ccc2cc(-c3ccc(OC)cc3)[nH]c2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.57
CASP3 P42574 2/20 0.57
SENP8 Q96LD8 2/20 0.57
SENP7 Q9BQF6 2/20 0.57
SENP6 Q9GZR1 2/20 0.57
KDM4E B2RXH2 2/20 0.57
NPC1 O15118 2/20 0.57
RAB9A P51151 2/20 0.57
CHEK2 O96017 1/20 0.55
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
ALDH1A1 P00352 3/20 0.50
KMT2A Q03164 2/20 0.50
MEN1 O00255 1/20 0.50
POLB P06746 1/20 0.50
KCNQ2 O43526 1/20 0.50
HPGD P15428 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
PRMT5 O14744 1/20 0.46
PRMT3 O60678 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5438780 0.88 CHEK2 (0.70) MAPTCASP3SENP8SENP7SENP6
SCHEMBL16329635 0.88 KDM4E (0.58) MAPTCASP3SENP8SENP7SENP6
SCHEMBL4880986 0.86 CASP3 (0.71) MAPTCASP3SENP8SENP7SENP6
SCHEMBL15223729 0.84 KDM4E (0.55) MAPTCASP3SENP8SENP7SENP6
SCHEMBL12392449 0.84 KDM4E (0.55) MAPTCASP3SENP8SENP7SENP6
SCHEMBL7945775 0.81 KDM4E (0.73) MAPTCASP3SENP8SENP7SENP6
SCHEMBL9132278 0.79 RARB (0.54) CASP3SENP8SENP7SENP6CHEK2
SCHEMBL28580125 0.79 RAB9A (0.61) MAPTCASP3SENP8SENP7SENP6
SCHEMBL30698055 0.78 CA1 (0.65) MAPTKDM4ECA1CA2KMT2A
SCHEMBL5606006 0.78 CA1 (0.65) MAPTKDM4ECA1CA2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070072911-A1 Indoles and azaindoles as antiviral agents AVOLIO SALVATORE 2007-03-29 US disclosed
EP-1673081-A1 INDOLES AND AZAINDOLES AS ANTIVIRAL AGENTS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2006-06-28 EP disclosed
WO-2005034941-A1 INDOLES AND AZAINDOLES AS ANTIVIRAL AGENTS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P ANGELETTI SPA (IT) 2005-04-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070072911-A1 Indoles and azaindoles as antiviral agents IDO1, IDO2, NAT1 MAPT 4298/4885CASP3 1343/4885SENP8 4535/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.