SCHEMBL5467716

SCHEMBL5467716

O=c1ccc2c(NCC(O)(CC3CCCc4cc(F)ccc43)C(F)(F)F)cccc2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 8/20 0.44
TRPV1 Q8NER1 6/20 0.38
PGR P06401 1/20 0.37
AR P10275 1/20 0.37
HTR6 P50406 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5470506 0.83 KDM4C (0.40) HTR6
SCHEMBL5475334 0.79 NR3C1 (0.38) NR3C1TRPV1PGRAR
SCHEMBL5474490 0.79 TRPV1 (0.37) NR3C1TRPV1PGRAR
SCHEMBL5471947 0.78 NR3C1 (0.41) NR3C1HTR6
SCHEMBL5471938 0.78 NR3C1 (0.41) NR3C1HTR6
SCHEMBL5471945 0.78 NR3C1 (0.41) NR3C1HTR6
SCHEMBL4827191 0.74 NR3C1 (0.68) NR3C1TRPV1PGR
SCHEMBL3650328 0.73 NR3C1 (0.67) NR3C1PGR
SCHEMBL5172786 0.71 NR3C1 (0.62) NR3C1PGR
SCHEMBL31390423 0.71 NR3C1 (0.57) NR3C1PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070129358-A1 Sbstituted chroman derivatives, processes for their preparation and their use as antiinflammatory agents SCHERING AG (DE) 2007-06-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070129358-A1 Sbstituted chroman derivatives, processes for their preparation and their use as antiinflammatory agents TNF, CXCL8, MPO NR3C1 83/4885TRPV1 1347/4885PGR 716/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.