SCHEMBL547293

SCHEMBL547293

CCC(=O)Oc1ccc2c(c1)CC[C@@H]1[C@@H]2CC[C@]2(C)[C@@H](O)CC[C@@H]12

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.80
ESR1 P03372 5/20 0.80
SMN1; SMN2 Q16637 4/20 0.80
ADORA3 P0DMS8 2/20 0.80
ATM Q13315 2/20 0.80
PGR P06401 2/20 0.80
AR P10275 2/20 0.80
SLC6A3 Q01959 2/20 0.80
CHRM1 P11229 1/20 0.80
TBXA2R P21731 1/20 0.80
ADRA1A P35348 1/20 0.80
OPRM1 P35372 1/20 0.80
MAPT P10636 5/20 0.79
KMT2A Q03164 4/20 0.79
MEN1 O00255 3/20 0.79
THRB P10828 1/20 0.79
NR3C1 P04150 2/20 0.73
SHBG P04278 2/20 0.73
SLC6A4 P31645 2/20 0.73
HTR2B P41595 2/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9404736 0.92 LMNA (0.77) LMNAESR1SMN1; SMN2ADORA3ATM
SCHEMBL4333126 0.91 LMNA (0.75) LMNAESR1SMN1; SMN2ADORA3ATM
SCHEMBL11102416 0.91 LMNA (0.75) LMNAESR1SMN1; SMN2ADORA3ATM
SCHEMBL40564 0.91 LMNA (0.75) LMNAESR1SMN1; SMN2ADORA3ATM
SCHEMBL14598803 0.91 LMNA (0.78) LMNAESR1SMN1; SMN2ADORA3ATM
Estradiol Dipropionate SCHEMBL5487956 0.91 MAPT (0.85) LMNAESR1SMN1; SMN2ADORA3ATM
SCHEMBL28077837 0.90 ESR1 (0.77) LMNAESR1SMN1; SMN2ADORA3ATM
SCHEMBL28792822 0.90 LMNA (0.86) LMNAESR1SMN1; SMN2ADORA3ATM
SCHEMBL547938 0.90 LMNA (0.73) LMNAESR1SMN1; SMN2ADORA3ATM
SCHEMBL1315380 0.90 LMNA (0.73) LMNAESR1SMN1; SMN2ADORA3ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 186 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180171288-A1 METHODS OF TREATING CANCER UNIVERSITY OF ROCHESTER 2018-06-21 US claimed
EP-1406633-B1 ENHANCED DRUG DELIVERY IN TRANSDERMAL SYSTEMS NOVEN PHARMA (US) 2011-10-05 EP claimed
US-20110097405-A1 ESTRADIOL-CONTAINING DRUG DELIVERY SYSTEM BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2011-04-28 US claimed
US-7846916-B2 Enhanced drug delivery in transdermal systems Noven Pharamaceticals, Inc. (US) 2010-12-07 US claimed
EP-2249803-A2 ESTRADIOL-CONTAINING DRUG DELIVERY SYSTEM Bayer Schering Pharma Aktiengesellschaft (DE) 2010-11-17 EP claimed
WO-2009101021-A2 ESTRADIOL-CONTAINING DRUG DELIVERY SYSTEM BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-08-20 WO claimed
EP-1814526-A2 ORAL SOLID DOSAGE FORMS CONTAINING A LOW DOSE OF ESTRADIOL Bayer Schering Pharma Aktiengesellschaft (DE) 2007-08-08 EP claimed
US-20060111334-A1 Oral solid dosage forms containing a low dose of estradiol BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2006-05-25 US claimed
WO-2006048261-A2 ORAL SOLID DOSAGE FORMS CONTAINING A LOW DOSE OF ESTRADIOL BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2006-05-11 WO claimed
US-20040209856-A1 Oral pharmaceutical products containing 17beta-estradiol-3-lower alkanoate, method of administering the same and process of preparation GALEN (CHEMICALS) LIMITED (IE) 2004-10-21 US claimed
US-5200197-A Contraceptive pill ALZA CORPORATION (US) 1993-04-06 US claimed
EP-0256668-B1 METHOD FOR TREATING MALE SEXUAL DYSFUNCTION UNIVERSITY OF FLORIDA (US) 1992-11-04 EP claimed
EP-0500793-A1 OSMOTIC, ORAL DOSAGE FORM FOR FERTILITY CONTROL. ALZA CORP (US) 1992-09-02 EP claimed
US-5098714-A OSMOTIC, ORAL DOSAGE FORM FOR FERTILITY CONTROL ALZA CORPORATION (US) 1992-03-24 US claimed
WO-1991007173-A1 OSMOTIC, ORAL DOSAGE FORM FOR FERTILITY CONTROL ALZA CORPORATION (US) 1991-05-30 WO claimed
US-4948593-A SUSTAINED AND CONTROLLED CONTRACEPTION ALZA CORPORATION (US) 1990-08-14 US claimed
US-4863911-A Method for treating male sexual dysfunction UNIVERSITY OF FLORIDA (US) 1989-09-05 US claimed
EP-0256668-A2 Method for treating male sexual dysfunction UNIVERSITY OF FLORIDA (US) 1988-02-24 EP claimed
EP-0220844-A2 Use of estrogen-dihydropyridine compounds for weight control UNIVERSITY OF FLORIDA (US) 1987-05-06 EP claimed
US-4617298-A STEROIDS UNIVERSITY OF FLORIDA (US) 1986-10-14 US claimed