Penmesterol

Penmesterol

SCHEMBL547668

C[C@]12CCC(OC3CCCC3)=CC1=CC[C@@H]1[C@@H]2CC[C@@]2(C)[C@H]1CC[C@]2(C)O

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SHBG P04278 2/20 0.48
ESR1 P03372 4/20 0.47
AR P10275 4/20 0.47
ESR2 Q92731 4/20 0.47
ALDH1A1 P00352 1/20 0.45
NR3C1 P04150 1/20 0.45
PGR P06401 1/20 0.45
ADRA1A P35348 1/20 0.45
HTR2B P41595 1/20 0.45
CYP2C19 P33261 1/20 0.43
SRD5A2 P31213 5/20 0.39
SRD5A1 P18405 2/20 0.39
CYP19A1 P11511 5/20 0.38
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pentagestrone SCHEMBL146311 0.87 SHBG (0.53) SHBGESR1ARESR2ALDH1A1
Pentagestrone SCHEMBL21405771 0.85 SHBG (0.51) SHBGESR1ARESR2ALDH1A1
SCHEMBL28118290 0.83 SHBG (0.49) SHBGESR1ARESR2ALDH1A1
SCHEMBL28118289 0.83 SHBG (0.49) SHBGESR1ARESR2ALDH1A1
SCHEMBL21405769 0.82 PGR (0.52) SHBGESR1ARESR2ALDH1A1
Quingestrone SCHEMBL145789 0.79 SRD5A2 (0.58) SHBGARALDH1A1NR3C1PGR
SCHEMBL9543900 0.77 SHBG (0.49) SHBGESR1ARESR2ALDH1A1
SCHEMBL11517207 0.74 CYP19A1 (0.64) SHBGESR1ARESR2ALDH1A1
SCHEMBL12178073 0.74 CYP19A1 (0.64) SHBGESR1ARESR2ALDH1A1
SCHEMBL28117758 0.74 CYP19A1 (0.64) SHBGESR1ARESR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 184 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-8110565-B2 Of the ACE inhibitor ramipril; controlling the melting point by mixing with the free acid with the ramipril ethyl or methyl ester prodrug and a pressure sensitive adhesive carrier; improved pharmacokinetics; sustained release NOVEN PHARMACEUTICALS, INC. (US) 2012-02-07 US claimed
EP-1406633-B1 ENHANCED DRUG DELIVERY IN TRANSDERMAL SYSTEMS NOVEN PHARMA (US) 2011-10-05 EP claimed
US-7879831-B2 Steroid on carrier containing pressure sensitive adhesive NOVEN PHARMACEUTICALS, INC. (US) 2011-02-01 US claimed
US-7867986-B2 Enhanced drug delivery in transdermal systems NOVEN PHARMACEUTICALS, INC. (US) 2011-01-11 US claimed
US-7846916-B2 Enhanced drug delivery in transdermal systems Noven Pharamaceticals, Inc. (US) 2010-12-07 US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
US-20080167280-A1 Enhanced drug delivery in transdermal systems NOVEN PHARMACEUTICALS, INC. 2008-07-10 US claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
US-20030232073-A1 Enhanced drug delivery in transdermal systems NOVEN PHARMACEUTICALS, INC. 2003-12-18 US claimed
US-20030152615-A1 Enhanced drug delivery in transdermal systems NOVEN PHARMACEUTICALS, INC. 2003-08-14 US claimed
US-20030152613-A1 Enhanced drug delivery in transdermal systems NOVEN PHARMACEUTICALS, INC. 2003-08-14 US claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
US-5656286-A BLEND OF TWO POLYMERS; PRESSURE SENSITIVE ADHESIVE NOVEN PHARMACEUTICALS, INC. (US) 1997-08-12 US claimed
EP-0496520-A1 Novel bone acting agents MERCK & CO. INC. (US) 1992-07-29 EP claimed
US-20250281509-A1 SEQUENTIAL HORMONE THERAPY TO IMPROVE SURVIVAL AND ENHANCE RESPONSE TO IMMUNE THERAPY IN MEN WITH PROSTATE CANCER THE JOHNS HOPKINS UNIVERSTY 2025-09-11 US disclosed
EP-0496520-A1 Novel bone acting agents MERCK & CO. INC. (US) 1992-07-29 EP disclosed