Pentagestrone

Pentagestrone

SCHEMBL146311

CC(=O)[C@@]1(O)CC[C@H]2[C@@H]3CC=C4C=C(OC5CCCC5)CC[C@]4(C)[C@H]3CC[C@@]21C

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SHBG P04278 3/20 0.53
LMNA P02545 4/20 0.50
CYP2C19 P33261 3/20 0.50
MEN1 O00255 2/20 0.50
NR3C1 P04150 2/20 0.50
MAPT P10636 2/20 0.50
KMT2A Q03164 2/20 0.50
SERPINA6 P08185 2/20 0.50
BLM P54132 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
ADORA3 P0DMS8 1/20 0.50
MAPK3 P27361 1/20 0.50
SLC6A3 Q01959 1/20 0.50
HIF1A Q16665 5/20 0.48
AR P10275 2/20 0.42
PGR P06401 1/20 0.42
CHRM1 P11229 1/20 0.42
SRD5A2 P31213 5/20 0.41
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pentagestrone SCHEMBL21405771 0.98 SHBG (0.51) SHBGLMNACYP2C19MEN1NR3C1
SCHEMBL11208571 0.88 LMNA (0.56) SHBGLMNACYP2C19MEN1NR3C1
Penmesterol SCHEMBL547668 0.87 SHBG (0.48) SHBGLMNACYP2C19NR3C1MAPT
SCHEMBL21405769 0.86 PGR (0.52) SHBGLMNACYP2C19MEN1NR3C1
SCHEMBL11517418 0.82 SHBG (0.59) SHBGLMNACYP2C19MEN1NR3C1
Quingestrone SCHEMBL145789 0.80 SRD5A2 (0.58) SHBGLMNACYP2C19MEN1NR3C1
SCHEMBL24358655 0.79 SHBG (0.53) SHBGLMNACYP2C19MEN1NR3C1
SCHEMBL9195965 0.79 SHBG (0.53) SHBGLMNACYP2C19MEN1NR3C1
SCHEMBL24358654 0.79 SHBG (0.53) SHBGLMNACYP2C19MEN1NR3C1
SCHEMBL11514918 0.77 SHBG (0.60) SHBGLMNACYP2C19MEN1NR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 437 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160008376-A1 Compositions, Methods and Uses for Treating Gender-Biased Immune Disorders BIOCOPEA LIMITED (GB) 2016-01-14 US claimed
WO-2016005599-A1 COMPOSITIONS, METHODS AND USES FOR TREATING GENDER-BIASED IMMUNE DISORDERS BIOCOPEA LIMITED (GB) 2016-01-14 WO claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
CN-101883556-B Transdermal delivery system for hormones and steroids ACRUX DDS PTY LTD 2013-05-29 CN claimed
US-8110565-B2 Of the ACE inhibitor ramipril; controlling the melting point by mixing with the free acid with the ramipril ethyl or methyl ester prodrug and a pressure sensitive adhesive carrier; improved pharmacokinetics; sustained release NOVEN PHARMACEUTICALS, INC. (US) 2012-02-07 US claimed
EP-1406633-B1 ENHANCED DRUG DELIVERY IN TRANSDERMAL SYSTEMS NOVEN PHARMA (US) 2011-10-05 EP claimed
US-20110195114-A1 TRANSDERMAL DELIVERY SYSTEMS FOR ACTIVE AGENTS ANTARES PHARMA, IPL, AG 2011-08-11 US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
US-7456159-B2 Enhanced drug delivery in transdermal systems NOVEN PHARMACEUTICALS, INC. (US) 2008-11-25 US claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
US-20030232073-A1 Enhanced drug delivery in transdermal systems NOVEN PHARMACEUTICALS, INC. 2003-12-18 US claimed
US-20030152614-A1 Enhanced drug delivery in transdermal systems NOVEN PHARMACEUTICALS, INC. 2003-08-14 US claimed
US-20030152615-A1 Enhanced drug delivery in transdermal systems NOVEN PHARMACEUTICALS, INC. 2003-08-14 US claimed
US-20030152613-A1 Enhanced drug delivery in transdermal systems NOVEN PHARMACEUTICALS, INC. 2003-08-14 US claimed
WO-2002102390-A1 ENHANCED DRUG DELIVERY IN TRANSDERMAL SYSTEMS NOVEN PHARMACEUTICALS, INC. (US) 2002-12-27 WO claimed
CN-1294519-A Pharmaceutical composition containing a compound having an activity of promoting the absorption of an active ingredient INPHARMA SA (CH) 2001-05-09 CN claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
EP-0496520-A1 Novel bone acting agents MERCK & CO. INC. (US) 1992-07-29 EP claimed
US-4016270-A Method for treating dysmenorrhea with a uterine therapeutic system ALZA CORPORATION (US) 1977-04-05 US claimed