SCHEMBL5482788

SCHEMBL5482788

O=C(N[C@@H](CC1CCCCC1)C(=O)NCC1CN(S(=O)(=O)c2ccc(Cl)cc2)CCO1)c1cc2ccccc2s1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
NPY5R Q15761 1/20 0.43
CCR1 P32246 1/20 0.42
UTS2R Q9UKP6 1/20 0.41
TACR2 P21452 5/20 0.41
REN P00797 1/20 0.39
PPM1D O15297 1/20 0.39
MMP1 P03956 2/20 0.39
MMP2 P08253 2/20 0.39
MMP3 P08254 2/20 0.39
TRPV4 Q9HBA0 2/20 0.38
CTSB P07858 1/20 0.38
CTSS P25774 1/20 0.38
MAPK1 P28482 1/20 0.38
CTSK P43235 1/20 0.38
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4179196 0.94 TACR2 (0.44) NPY5RUTS2RTACR2RENCTSB
SCHEMBL4192205 0.91 TRPV4 (0.47) KMT2AMEN1CCR1TACR2REN
SCHEMBL4178416 0.89 UTS2R (0.51) KMT2AMEN1NPY5RCCR1UTS2R
SCHEMBL4175710 0.88 CTSK (0.44) KMT2AMEN1NPY5RCCR1UTS2R
SCHEMBL4188403 0.88 MAPK1 (0.49) KMT2AMEN1NPY5RCCR1UTS2R
SCHEMBL4181435 0.87 CCR1 (0.46) KMT2AMEN1NPY5RCCR1UTS2R
SCHEMBL4181213 0.86 CTSL (0.50) KMT2AMEN1MMP1MMP2MMP3
SCHEMBL4191791 0.86 CTSB (0.42) UTS2RTACR2RENCTSBCTSS
SCHEMBL4180771 0.84 CCR1 (0.47) KMT2AMEN1NPY5RCCR1UTS2R
SCHEMBL4194752 0.83 CTSK (0.51) UTS2RTACR2CTSBCTSSMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1869026-A1 NOVEL COMPOUNDS SmithKline Beecham Corporation (US) 2007-12-26 EP disclosed
WO-2006105475-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-10-05 WO disclosed