SCHEMBL5486374

SCHEMBL5486374

CCCCCn1nc[nH]c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 2/20 0.42
PTGS1 P23219 3/20 0.40
PTGS2 P35354 3/20 0.40
MGLL Q99685 2/20 0.40
FAAH O00519 1/20 0.40
PDE4A P27815 2/20 0.39
ADORA2A P29274 2/20 0.39
PDE4B Q07343 2/20 0.39
PDE4C Q08493 2/20 0.39
PDE4D Q08499 2/20 0.39
ADORA3 P0DMS8 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.39
HSP90AA1 P07900 1/20 0.39
CYP3A4 P08684 1/20 0.39
G6PD P11413 1/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
HIF1A Q16665 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2826206 0.98 ADORA2B (0.44) ADORA2BPTGS1PTGS2MGLLFAAH
SCHEMBL1723957 0.94 ADORA2A (0.43) ADORA2BPDE4AADORA2APDE4BPDE4C
SCHEMBL22944867 0.86
SCHEMBL16325249 0.79 SLC9A1 (0.38) ADORA2BPTGS1PTGS2MGLLFAAH
SCHEMBL18713930 0.78 SLC9A1 (0.39) ADORA2BPTGS1PTGS2MGLLFAAH
SCHEMBL31330275 0.77 ADORA2A (0.31) ADORA2BADORA2A
SCHEMBL31330320 0.75 ADORA3 (0.32) ADORA2BADORA3
SCHEMBL6268666 0.75 PDE3A (0.47) PTGS1PTGS2MGLLFAAHCYP1A2
SCHEMBL31330313 0.74 ADORA2A (0.33) ADORA2BADORA2AALDH1A1
SCHEMBL31330327 0.74 ADORA2A (0.33) ADORA2BPDE4AADORA2APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 88 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0831705-B1 N-ARYL-1,2,4-TRIAZOLIN-5-ONES BAYER AG (DE) 2001-08-29 EP claimed
EP-0942907-A1 2R, 4S, S, R- AND 2S, 4R, S, R-HYDROXYITRACONAZOLE SEPRACOR, INC. (US) 1999-09-22 EP claimed
EP-0938484-A1 2R,4S,R,R- AND 2S,4R,R,R-HYDROXYITRACONAZOLE SEPRACOR, INC. (US) 1999-09-01 EP claimed
EP-0938487-A2 2$i(R),4$i(S),$i(R),$i(S)- AND 2$i(S),4$i(R),$i(R),$i(S)-HYDROXYITRACONAZOLE- AND HYDROXYSAPERCONAZOLE DERIVATIVES SEPRACOR, INC. (US) 1999-09-01 EP claimed
EP-0937071-A1 2R,4S,S,S- AND 2S,4R,S,S-HYDROXYITRACONAZOLE SEPRACOR, INC. (US) 1999-08-25 EP claimed
WO-1998021213-A2 2R,4S,R,S- AND 2S,4R,R,S-HYDROXYITRACONAZOLE- AND HYDROXYSAPERCONAZOLE DERIVATIVES SEPRACOR, INC. (US) 1998-05-22 WO claimed
WO-1998021205-A1 2R,4S,R,R- AND 2S,4R,R,R-HYDROXYITRACONAZOLE SEPRACOR, INC. (US) 1998-05-22 WO claimed
WO-1998021204-A1 2R,4S,S,S- AND 2S,4R,S,S-HYDROXYITRACONAZOLE SEPRACOR, INC. (US) 1998-05-22 WO claimed
WO-1998021203-A1 2R,4S,S,R- AND 2S,4R,S,R-HYDROXYITRACONAZOLE SEPRACOR, INC. (US) 1998-05-22 WO claimed
EP-0831705-A1 N-ARYL-1,2,4-TRIAZOLIN-5-ONES BAYER AG (DE) 1998-04-01 EP claimed
WO-1996041535-A1 N-ARYL-1,2,4-TRIAZOLIN-5-ONES BAYER AKTIENGESELLSCHAFT (DE) 1996-12-27 WO claimed
EP-0221083-A1 HALOALKYL TRIAZOLINONES FMC Corporation (US) 1987-05-13 EP claimed
WO-1986004481-A2 HALOALKYL TRIAZOLINONES FMC CORPORATION (US) 1986-08-14 WO claimed
WO-2024249959-A1 COMPOSITIONS REDUCING THE EXPRESSION OR ACTIVITY OF C1 GALT1 FOR TREATING EWING SARCOMA UNIVERSITY OF MASSACHUSETTS MEDICAL SCHOOL (US) 2024-12-05 WO disclosed
US-9981940-B2 Aryl sulfide derivatives and aryl sulfoxide derivatives as acaricides and insecticides BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2018-05-29 US disclosed
CN-104672157-B A kind of preparation method of aryltriazolinones 山东潍坊润丰化工股份有限公司 2017-06-27 CN disclosed
EP-0221083-A1 HALOALKYL TRIAZOLINONES FMC Corporation (US) 1987-05-13 EP disclosed
EP-0221083-A1 HALOALKYL TRIAZOLINONES FMC Corporation (US) 1987-05-13 EP disclosed
WO-1986004481-A2 HALOALKYL TRIAZOLINONES FMC CORPORATION (US) 1986-08-14 WO disclosed
WO-1986004481-A2 HALOALKYL TRIAZOLINONES FMC CORPORATION (US) 1986-08-14 WO disclosed