SCHEMBL1723957

SCHEMBL1723957

CCCCn1nc[nH]c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 8/20 0.43
PDE4A P27815 7/20 0.43
PDE4B Q07343 7/20 0.43
PDE4C Q08493 7/20 0.43
PDE4D Q08499 7/20 0.43
ADORA2B P29275 6/20 0.43
ADORA3 P0DMS8 3/20 0.43
TOP2A P11388 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
KMT2A Q03164 1/20 0.36
ADORA1 P30542 2/20 0.35
SLC9A1 P19634 1/20 0.35
HPGD P15428 1/20 0.35
BLM P54132 1/20 0.35
PDE3A Q14432 1/20 0.35
HSD17B10 Q99714 1/20 0.35
BRD4 O60885 1/20 0.35
BRD2 P25440 1/20 0.35
BRD3 Q15059 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5486374 0.94 ADORA2B (0.42) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL2826206 0.93 ADORA2B (0.44) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL22944867 0.88
SCHEMBL31330320 0.77 ADORA3 (0.32) ADORA2BADORA3
SCHEMBL31330313 0.75 ADORA2A (0.33) ADORA2AADORA2BALDH1A1ADORA1
SCHEMBL31330327 0.75 ADORA2A (0.33) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL31330241 0.75 ADORA2A (0.33) ADORA2AADORA2BALDH1A1ADORA1
SCHEMBL31330275 0.75 ADORA2A (0.31) ADORA2AADORA2BADORA1
SCHEMBL18462236 0.74 DAO (0.48) PDE4APDE4BPDE4CPDE4DADORA2B
SCHEMBL16325249 0.73 SLC9A1 (0.38) ADORA2BALDH1A1KMT2ASLC9A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024249959-A1 COMPOSITIONS REDUCING THE EXPRESSION OR ACTIVITY OF C1 GALT1 FOR TREATING EWING SARCOMA UNIVERSITY OF MASSACHUSETTS MEDICAL SCHOOL (US) 2024-12-05 WO disclosed
EP-3356362-B1 2-(HET)ARYL-SUBSTITUTED CONDENSED HETEROCYCLIC DERIVATIVES USEFUL AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2021-02-03 EP disclosed
CN-102333779-B Benzopyran and benzoxex PI3K inhibitor compounds and methods of use GENENTECH, INC. (US) 2015-12-09 CN disclosed
EP-2343980-A1 TRIAZOLE ANTIFUNGAL AGENTS Wu, Nian (US) 2011-07-20 EP disclosed
WO-2010027496-A1 TRIAZOLE ANTIFUNGAL AGENTS WU NIAN (US) 2010-03-11 WO disclosed