SCHEMBL5487538

SCHEMBL5487538

c1ccc(-c2cccc(COCc3cccc(-c4ccccc4)c3N3CCCC3)c2N2CCCC2)cc1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 5/20 0.41
TACR1 P25103 1/20 0.40
CHRNB2 P17787 2/20 0.40
CHRNA4 P43681 2/20 0.40
CD274 Q9NZQ7 7/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
PRKDC P78527 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
DPP4 P27487 1/20 0.37
PDCD1 Q15116 1/20 0.37
TSHR P16473 1/20 0.36
RECQL P46063 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20360396 0.81 ALDH1A1 (0.46) HTR7PRKDCKDM4EALDH1A1TDP1
SCHEMBL20360705 0.79 PRKDC (0.48) HTR7PRKDCKDM4EALDH1A1TDP1
SCHEMBL336977 0.73 TACR1 (0.62) HTR7TACR1CHRNB2CHRNA4CD274
SCHEMBL9338655 0.70 TACR1 (0.58) HTR7TACR1CHRNB2CHRNA4CD274
SCHEMBL27844226 0.69 CD274 (0.67) TACR1CD274PDCD1
SCHEMBL8679174 0.67 TACR1 (0.51) HTR7TACR1CHRNB2CHRNA4CD274
SCHEMBL16390993 0.67 TACR1 (0.64) TACR1CHRNB2CHRNA4CD274CHRNB4
SCHEMBL10599800 0.67 TACR1 (0.64) TACR1CHRNB2CHRNA4CD274CHRNB4
SCHEMBL18181830 0.67 TACR1 (0.48) TACR1CHRNB2CHRNA4CD274ALDH1A1
SCHEMBL483515 0.67 PTGS2 (0.52) HTR7ALDH1A1L3MBTL1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101142181-B Process for the preparation of enantiomerically pure 4-pyrrolidinophenylbenzyl ether derivatives HOFFMANN LA ROCHE 2011-05-04 CN disclosed
CN-101142181-A Process for the preparation of enantiomerically pure 4-pyrrolidinophenylbenzyl ether derivatives HOFFMANN LA ROCHE (CH) 2008-03-12 CN disclosed
EP-1861362-A1 METHOD FOR PREPARING ENANTIOMERICALLY PURE 4-PYRROLIDINOPHENYL, BENZYL, ETHER DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2007-12-05 EP disclosed
WO-2006097197-A1 METHOD FOR PREPARING ENANTIOMERICALLY PURE 4-PYRROLIDINOPHENYL, BENZYL, ETHER DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2006-09-21 WO disclosed