Histidine

Histidine

SCHEMBL5491748

NC1CCCCC1.N[C@@H](Cc1c[nH]cn1)C(=O)O

nearest known ligand 0.38

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP1A2 P05177 1/20 0.37
TPH1 P17752 2/20 0.36
CPB2 Q96IY4 4/20 0.34
KIF11 P52732 1/20 0.34
ALPI P09923 1/20 0.33
PKM P14618 1/20 0.33
PTGS1 P23219 1/20 0.33
XIAP P98170 1/20 0.33
GRIK1 P39086 1/20 0.33
CPB1 P15086 1/20 0.33
GRIA1 P42261 1/20 0.33
GRIA2 P42262 1/20 0.33
GRIA3 P42263 1/20 0.33
GRIA4 P48058 1/20 0.33
GRIN2D O15399 5/20 0.32
GRIN3B O60391 5/20 0.32
GRIN1 Q05586 5/20 0.32
GRIN2A Q12879 5/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Histidine SCHEMBL5491744 1.00 SLC7A5 (0.38) SLC7A5CYP3A4CYP1A2TPH1CPB2
Histidine SCHEMBL27762881 0.87 TPH1 (0.38) SLC7A5CYP3A4CYP1A2TPH1CPB2
Histidine SCHEMBL3258 0.86 SLC7A5 (0.47) SLC7A5CYP3A4CYP1A2ALPIPKM
Histidine SCHEMBL163443 0.86 SLC7A5 (0.47) SLC7A5CYP3A4CYP1A2ALPIPKM
Histidine SCHEMBL3259 0.86 SLC7A5 (0.47) SLC7A5CYP3A4CYP1A2ALPIPKM
Histidine SCHEMBL18824897 0.86 SLC7A5 (0.47) SLC7A5CYP3A4CYP1A2ALPIPKM
Histidine SCHEMBL388563 0.86 SLC7A5 (0.47) SLC7A5CYP3A4CYP1A2ALPIPKM
Histidine SCHEMBL163442 0.86 SLC7A5 (0.47) SLC7A5CYP3A4CYP1A2ALPIPKM
Histidine SCHEMBL995910 0.86 SLC7A5 (0.47) SLC7A5CYP3A4CYP1A2ALPIPKM
Histidine SCHEMBL8080341 0.86 SLC7A5 (0.47) SLC7A5CYP3A4CYP1A2ALPIPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1858538-A2 MUCIN HYPERSECRETION INHIBITORS BASED ON THE STRUCTURE OF MANS AND METHODS OF USE Biomarck Pharmaceuticals, Ltd. (US) 2007-11-28 EP disclosed
WO-2006078899-A2 MUCIN HYPERSECRETION INHIBITORS BASED ON THE STRUCTURE OF MANS AND METHODS OF USE BIOMARCK PHARMACEUTICALS, LTD. (US) 2006-07-27 WO disclosed