SCHEMBL5491925

SCHEMBL5491925

CON(C(=O)c1ccc(-c2ccccc2)cc1Cc1ccccc1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 1/20 0.48
PTPN1 P18031 1/20 0.45
CNR1 P21554 2/20 0.43
CNR2 P34972 2/20 0.43
DCLRE1A Q6PJP8 1/20 0.42
DCLRE1B Q9H816 1/20 0.42
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
OXTR P30559 1/20 0.40
AVPR1A P37288 1/20 0.40
ESR1 P03372 1/20 0.39
CDC7 O00311 1/20 0.39
ROCK2 O75116 1/20 0.39
MAP4K4 O95819 1/20 0.39
GSK3B P49841 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1926265 0.78 PTPN1 (0.48) SLC6A9PTPN1CNR1CNR2DCLRE1A
SCHEMBL1927147 0.77 PTPN1 (0.52) SLC6A9PTPN1CNR1CNR2DCLRE1A
SCHEMBL1926320 0.73 PTPN1 (0.51) SLC6A9PTPN1CNR1CNR2DCLRE1A
SCHEMBL2595456 0.73 CDC25B (0.47) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL27929241 0.71 DCLRE1B (0.52) SLC6A9PTPN1CNR1CNR2DCLRE1A
SCHEMBL6489038 0.67 MAPT (0.51) PTPN1ALDH1A1MEN1MAPTKMT2A
SCHEMBL27542931 0.67 EGFR (0.52) DCLRE1ADCLRE1BALDH1A1KDM4EMEN1
SCHEMBL92795 0.67 MEN1 (0.54) SLC6A9DCLRE1ADCLRE1BALDH1A1KDM4E
SCHEMBL9517957 0.67 MAPT (0.47) PTPN1ALDH1A1KDM4EMEN1MAPT
SCHEMBL15940350 0.67 SLC6A9 (0.52) SLC6A9PTPN1ALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1763509-A1 ALPHA-HELICAL MIMETICS THE WALTER AND ELIZA HALL INSTITUTE OF MEDICAL RESEARCH (AU) 2007-03-21 EP disclosed
WO-2006002474-A1 ALPHA-HELICAL MIMETICS THE WALTER AND ELIZA HALL INSTITUTE OF MEDICAL RESEARCH (AU) 2006-01-12 WO disclosed