SCHEMBL5493797

SCHEMBL5493797

Cn1ncc(NC(=O)NCCNC(=O)O)c1NC(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 2/20 0.42
KMT2A Q03164 5/20 0.39
MEN1 O00255 3/20 0.39
MAPT P10636 3/20 0.39
ITGB3 P05106 2/20 0.39
ITGAV P06756 2/20 0.39
UTS2R Q9UKP6 1/20 0.37
LMNA P02545 2/20 0.36
POLB P06746 3/20 0.36
KDM4E B2RXH2 1/20 0.36
HTT P42858 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
EPHX1 P07099 1/20 0.36
TSHR P16473 1/20 0.35
ITGB1 P05556 1/20 0.35
ITGA5 P08648 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19213536 0.91 EPHX1 (0.46) NTRK1KMT2AMEN1MAPTITGB3
SCHEMBL5494715 0.90 ITGB3 (0.36) NTRK1KMT2AMAPTITGB3ITGAV
SCHEMBL5499949 0.90 KMT2A (0.36) NTRK1KMT2AMEN1MAPTLMNA
SCHEMBL5493399 0.90 NTRK1 (0.39) NTRK1KMT2AMEN1MAPTITGB3
Carbamic Acid SCHEMBL5493402 0.89 NTRK1 (0.40) NTRK1KMT2AMEN1MAPTITGB3
SCHEMBL5493337 0.89 CYP2C9 (0.37) NTRK1KMT2AKDM4ERAB9ATSHR
SCHEMBL19399313 0.88 NTRK1 (0.39) NTRK1KMT2AMEN1MAPTITGB3
SCHEMBL5492718 0.87 BCHE (0.40) NTRK1LMNAPOLB
SCHEMBL3121437 0.87 NTRK1 (0.36) NTRK1MAPTLMNASMN1; SMN2TSHR
SCHEMBL3123213 0.86 NTRK1 (0.35) NTRK1KMT2AMEN1MAPTUTS2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112321610-B Ceclozapine sulfate and preparation method and application thereof 湖南润星制药有限公司 2022-04-19 CN claimed
CN-112321610-A Ceclozapine sulfate and preparation method and application thereof 湖南润星制药有限公司 2021-02-05 CN claimed
EP-3468968-B1 SOLID FORMS OF CEFTOLOZANE AND PROCESSES FOR PREPARING MERCK SHARP & DOHME LLC (US) 2024-01-10 EP disclosed
US-11542279-B2 Solid forms of ceftolozane and processes for preparing MERCK SHARP & DOHME LLC (US) 2023-01-03 US disclosed
CN-112321610-B Ceclozapine sulfate and preparation method and application thereof 湖南润星制药有限公司 2022-04-19 CN disclosed
CN-112321610-B Ceclozapine sulfate and preparation method and application thereof 湖南润星制药有限公司 2022-04-19 CN disclosed
US-20220056045-A1 SOLID FORMS OF CEFTOLOZANE AND PROCESSES FOR PREPARING MERCK SHARP & DOHME CORP. (US) 2022-02-24 US disclosed
CN-112321610-A Ceclozapine sulfate and preparation method and application thereof 湖南润星制药有限公司 2021-02-05 CN disclosed
CN-112321610-A Ceclozapine sulfate and preparation method and application thereof 湖南润星制药有限公司 2021-02-05 CN disclosed
EP-3347362-B1 PROCESS FOR PREPARING CEFTOLOZANE FROM 7-AMINOCEPHALOSPORANIC ACID (7-ACA) SANDOZ AG (CH) 2019-10-23 EP disclosed
EP-3468968-A1 SOLID FORMS OF CEFTOLOZANE AND PROCESSES FOR PREPARING Merck Sharp & Dohme Corp. (US) 2019-04-17 EP disclosed
US-9006421-B2 Cephalosporin compositions and methods of manufacture CUBIST PHARMACEUTICALS, INC. (US) 2015-04-14 US disclosed
EP-1556389-B3 CEPHEM COMPOUNDS ASTELLAS PHARMA INC (JP) 2015-04-01 EP disclosed
WO-2014152763-A1 CEPHALOSPORIN COMPOSITIONS AND METHODS OF MANUFACTURE CUBIST PHARMACEUTICALS, INC. (US) 2014-09-25 WO disclosed
US-20140274958-A1 CEPHALOSPORIN COMPOSITIONS AND METHODS OF MANUFACTURE MERCK SHARP & DOHME LLC 2014-09-18 US disclosed
US-20140274999-A1 CEPHALOSPORIN COMPOSITIONS AND METHODS OF MANUFACTURE MERCK SHARP & DOHME CORP. 2014-09-18 US disclosed
EP-1556389-B1 CEPHEM COMPOUNDS ASTELLAS PHARMA INC (JP) 2007-07-25 EP disclosed
US-20070037786-A1 Cephem compounds WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 2007-02-15 US disclosed
US-7129232-B2 For therapy of of infectious diseases ASTELLAS PHARMA INC. (JP) 2006-10-31 US disclosed
US-20040132994-A1 Cephem compounds FUJISAWA PHARMACEUTICAL CO., LTD (JP) 2004-07-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070037786-A1 Cephem compounds CEP170, ABCB11, SLC7A1 NTRK1 2964/4885KMT2A 2510/4885MEN1 651/4885
US-20040132994-A1 Cephem compounds CEP170, ABCB11, RCC2 NTRK1 3809/4885KMT2A 2826/4885MEN1 868/4885
US-20140274999-A1 CEPHALOSPORIN COMPOSITIONS AND METHODS OF MANUFACTURE CYP3A7, SEPTIN7, PEPD NTRK1 4368/4885KMT2A 1025/4885MEN1 612/4885
US-20140274958-A1 CEPHALOSPORIN COMPOSITIONS AND METHODS OF MANUFACTURE CYP3A7, SEPTIN7, PEPD NTRK1 4368/4885KMT2A 1025/4885MEN1 612/4885
US-11542279-B2 Solid forms of ceftolozane and processes for preparing PPP1CC, CCNC, AMPD3 NTRK1 4563/4885KMT2A 1853/4885MEN1 2281/4885
US-20220056045-A1 SOLID FORMS OF CEFTOLOZANE AND PROCESSES FOR PREPARING PPP1CC, CCNC, AMPD3 NTRK1 4563/4885KMT2A 1853/4885MEN1 2281/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.