SCHEMBL5493891

SCHEMBL5493891

COC(=O)c1[c]cccc1-c1ccc(C(F)(F)F)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.43
PTPN1 P18031 1/20 0.41
SLC6A3 Q01959 3/20 0.41
SLC6A4 P31645 2/20 0.41
CFTR P13569 1/20 0.40
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
KLRK1 P26718 3/20 0.38
MICA Q29983 3/20 0.38
RAET1L Q5VY80 3/20 0.38
APP P05067 1/20 0.38
MAPK14 Q16539 1/20 0.38
MYC P01106 1/20 0.38
MAX P61244 1/20 0.38
TP53 P04637 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.37
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
KIF11 P52732 2/20 0.37
APOB P04114 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7820684 0.81 KDM4E (0.51) BACE1SLC6A3SLC6A4
SCHEMBL10645473 0.77 SLC6A3 (0.69) BACE1SLC6A3SLC6A4CFTRKLRK1
SCHEMBL29979725 0.77 SLC6A3 (0.69) BACE1SLC6A3SLC6A4CFTRKLRK1
SCHEMBL4285343 0.76 NOTUM (0.43) CFTR
SCHEMBL29917415 0.73 SLC6A3 (0.52) BACE1PTPN1SLC6A3SLC6A4CFTR
SCHEMBL30755410 0.73 BACE1 (0.44) BACE1PTPN1SLC6A3SLC6A4CFTR
SCHEMBL7041867 0.73 BACE1 (0.44) BACE1PTPN1SLC6A3SLC6A4CFTR
SCHEMBL28825335 0.72 KLRK1 (0.52) BACE1KLRK1MICARAET1L
SCHEMBL8728062 0.72 SLC6A3 (0.50) SLC6A3SLC6A4CFTRMYC
SCHEMBL9556244 0.71 SLC6A3 (0.41) PTPN1SLC6A3SLC6A4CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7304086-B2 Inhibitors of glutaminyl cyclase PROBIODRUG AG (DE) 2007-12-04 US claimed