SCHEMBL5498764

SCHEMBL5498764

CCCC(=O)Nc1ccc(Oc2ccc(C#N)c(Cl)c2)cc1.Cc1cc(F)ccc1Oc1ccc(C#N)c(Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AR P10275 2/20 0.49
MTNR1B P49286 4/20 0.47
MTNR1A P48039 3/20 0.46
PLA2G7 Q13093 4/20 0.44
ESRRA P11474 1/20 0.43
PFKFB2 O60825 3/20 0.42
PFKFB1 P16118 3/20 0.42
PFKFB3 Q16875 3/20 0.42
SLC22A12 Q96S37 3/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C8 P10632 1/20 0.41
KCNH2 Q12809 1/20 0.41
SLC22A6 Q4U2R8 1/20 0.41
SLC22A8 Q8TCC7 1/20 0.41
SLC22A11 Q9NSA0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4171293 0.87 MTNR1B (0.58) MTNR1BMTNR1APLA2G7ESRRAPFKFB2
SCHEMBL4181443 0.81 AR (0.72) ARSLC22A12CYP3A4CYP2C9CYP2C19
SCHEMBL17536366 0.76 MTNR1B (0.63) ARMTNR1BMTNR1APFKFB2PFKFB1
SCHEMBL17536369 0.75 MTNR1B (0.56) MTNR1BMTNR1APFKFB2PFKFB1PFKFB3
SCHEMBL8145133 0.72 MTNR1B (0.74) MTNR1BMTNR1A
SCHEMBL18615328 0.71 AR (0.60) ARPLA2G7SLC22A12
SCHEMBL4171343 0.70 AR (0.59) ARSLC22A12CYP3A4CYP2C9CYP2C19
SCHEMBL4163780 0.69 AR (0.72) ARESRRASLC22A12KCNH2
SCHEMBL4186077 0.69 AR (0.67) ARSLC22A12CYP3A4CYP2C9CYP2C19
SCHEMBL28913547 0.69 AR (0.57) ARPLA2G7SLC22A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781280-A2 ANDROGEN MODULATORS Warner-Lambert Company LLC (US) 2007-05-09 EP claimed
WO-2006018723-A2 ANDROGEN MODULATORS WARNER-LAMBERT COMPANY LLC (US) 2006-02-23 WO claimed