SCHEMBL5499016

SCHEMBL5499016

OC1(CCCc2cccc(OC(F)F)c2F)CCNCC1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.38
SLC6A2 P23975 7/20 0.38
SLC6A4 P31645 7/20 0.38
SLC6A3 Q01959 5/20 0.38
CYP2D6 P10635 2/20 0.37
SIGMAR1 Q99720 1/20 0.32
REN P00797 1/20 0.31
HTR1A P08908 2/20 0.31
OPRM1 P35372 1/20 0.30
OPRD1 P41143 1/20 0.30
OPRK1 P41145 1/20 0.30
OPRL1 P41146 1/20 0.30
TACR1 P25103 1/20 0.30
PIM1 P11309 1/20 0.30
PIM2 Q9P1W9 1/20 0.30
GPR4 P46093 1/20 0.30
USP2 O75604 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5494489 0.93 SLC6A2 (0.40) KCNH2SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL5495138 0.87 KCNH2 (0.37) KCNH2SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL5502120 0.83 SLC6A2 (0.38) KCNH2SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL4390004 0.81 FFAR4 (0.39) KCNH2SLC6A2SLC6A4SLC6A3SIGMAR1
SCHEMBL5501435 0.80 KCNH2 (0.38) KCNH2SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL5493818 0.79 FFAR4 (0.41) KCNH2SLC6A2SLC6A4SLC6A3REN
SCHEMBL2785289 0.77 FFAR4 (0.43) SLC6A2SLC6A4TACR1
SCHEMBL5502309 0.76 KCNH2 (0.38) KCNH2SLC6A2SLC6A4RENOPRM1
SCHEMBL5499318 0.74 KCNH2 (0.33) KCNH2SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL5495293 0.73 P2RX7 (0.38) KCNH2SLC6A2SLC6A4SLC6A3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765779-A1 NEW SUBSTITUTED PIPERIDINES AS MODULATORS OF DOPAMINE NEUROTRANSMISSION A. CARLSSON RESEARCH AB (SE) 2007-03-28 EP disclosed
WO-2005121092-A1 NEW SUBSTITUTED PIPERIDINES AS MODULATORS OF DOPAMINE NEUROTRANSMISSION A. CARLSSON RESEARCH AB (SE) 2005-12-22 WO disclosed