SCHEMBL5502292

SCHEMBL5502292

CC(C)c1c(N)cc2c(c1F)NC(=O)C2

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.32
TDP2 O95551 1/20 0.31
GRIA1 P42261 3/20 0.31
CACNG8 Q8WXS5 3/20 0.31
HDAC3 O15379 1/20 0.31
KDM5B Q9UGL1 1/20 0.31
MET P08581 1/20 0.30
SMYD3 Q9H7B4 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5504614 0.80 HDAC3 (0.35) AHRTDP2GRIA1CACNG8HDAC3
SCHEMBL5504827 0.77 TDP2 (0.36) TDP2GRIA1CACNG8
SCHEMBL5501936 0.76 AHR (0.32) AHRTDP2GRIA1CACNG8HDAC3
SCHEMBL5506392 0.74 GRM2 (0.36)
SCHEMBL5502598 0.74 AHR (0.30) AHRTDP2HDAC3
SCHEMBL5505582 0.73 EPHX2 (0.33) AHRTDP2GRIA1CACNG8HDAC3
SCHEMBL5498389 0.73 DRD2 (0.33) AHRTDP2GRIA1CACNG8HDAC3
SCHEMBL151642 0.70 HDAC3 (0.40) AHRTDP2GRIA1CACNG8HDAC3
SCHEMBL23612469 0.70 GRIA1 (0.39) AHRTDP2GRIA1CACNG8
SCHEMBL5507259 0.70 GRIN1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1869030-A1 7-FLUORO-1,3-DIHYDRO-INDOL-2-ONE OXAZOLIDINONES AS ANTIBACTERIAL AGENTS Pharmacia & Upjohn Company LLC (US) 2007-12-26 EP disclosed
EP-1781642-A1 OXAZOLIDINONES CONTAINING OXINDOLES AS ANTIBACTERIAL AGENTS Pharmacia & Upjohn Company LLC (US) 2007-05-09 EP disclosed
EP-1781643-A1 OXINDOLE OXAZOLIDINONES AS ANTIBACTERIAL AGENTS Pharmacia & Upjohn Company LLC (US) 2007-05-09 EP disclosed
WO-2006106427-A1 7-FLUORO-1,3-DIHYDRO-INDOL-2-ONE OXAZOLIDINONES AS ANTIBACTERIAL AGENTS PHARMACIA & UPJOHN COMPANY LLC (US) 2006-10-12 WO disclosed
WO-2006016221-A1 OXAZOLIDINONES CONTAINING OXINDOLES AS ANTIBACTERIAL AGENTS PHARMACIA & UPJOHN COMPANY LLC (US) 2006-02-16 WO disclosed
WO-2006016220-A1 OXINDOLE OXAZOLIDINONES AS ANTIBACTERIAL AGENTS PHARMACIA & UPJOHN COMPANY LLC (US) 2006-02-16 WO disclosed