SCHEMBL5503490

SCHEMBL5503490

CC(C)Cn1c(N)nc2[nH]cnc2c1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.49
ADORA2B P29275 4/20 0.49
PDE2A O00408 6/20 0.47
PDE1A P54750 4/20 0.47
PDE1B Q01064 4/20 0.47
PDE1C Q14123 4/20 0.47
CFTR P13569 2/20 0.47
PDE5A O76074 2/20 0.47
PDE4A P27815 2/20 0.47
PDE4B Q07343 2/20 0.47
PDE4C Q08493 2/20 0.47
PDE4D Q08499 2/20 0.47
ADORA1 P30542 2/20 0.47
TSHR P16473 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
MAPK1 P28482 1/20 0.47
SCN1A P35498 1/20 0.47
PDE6C P51160 1/20 0.47
PDE3B Q13370 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL874734 0.84 ADORA2A (0.45) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL17186378 0.83 PNP (0.39) ADORA2AADORA2BPDE2APDE1APDE1B
SCHEMBL18605634 0.83 PNP (0.39) ADORA2AADORA2BPDE2APDE1APDE1B
SCHEMBL9960806 0.83 PNP (0.38) ADORA2AADORA2BPDE4APDE4BPDE4C
Hydrochloric Acid SCHEMBL17186422 0.82 PNP (0.39) ADORA2AADORA2BPDE2APDE1APDE1B
SCHEMBL21748352 0.82 ADORA2A (0.40) ADORA2AADORA2BADORA1SMN1; SMN2PNP
SCHEMBL6268075 0.81 ADORA2A (0.34) ADORA2AADORA2BPDE2APDE1APDE1B
SCHEMBL667794 0.81 PDE4A (0.49) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL6271387 0.80 CDK1 (0.37) ADORA2AADORA2BPDE2APDE1APDE1B
SCHEMBL2113436 0.80 ADORA2A (0.33) ADORA2AADORA2BPDE2APDE1APDE1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0977767-B1 AMINOOXY-MODIFIED OLIGONUCLEOTIDES ISIS PHARMACEUTICALS INC (US) 2007-09-19 EP claimed
JP-60199899-A None JP disclosed
JP-S60199899-A NUCLEOSIDE 3'-PHOSPHOTRIESTER DERIVATIVE FUJIREBIO INC 1985-10-09 JP disclosed