SCHEMBL874734

SCHEMBL874734

CCn1c(N)nc2[nH]cnc2c1=O

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 14/20 0.45
ADORA2B P29275 8/20 0.45
PDE4A P27815 13/20 0.44
PDE4B Q07343 13/20 0.44
PDE4C Q08493 13/20 0.44
PDE4D Q08499 13/20 0.44
TSHR P16473 1/20 0.38
ADORA3 P0DMS8 2/20 0.36
PNP P00491 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL667794 0.88 PDE4A (0.49) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL9960806 0.87 PNP (0.38) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL6272726 0.85 PDE4A (0.49) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL1767742 0.84 ADORA2A (0.39) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL8522266 0.84 ADORA2B (0.51) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL5503490 0.84 ADORA2A (0.49) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL8536000 0.83 ADORA2B (0.53) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL6272293 0.83 ADORA2B (0.53) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL4384737 0.83 ADORA2B (0.53) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL6265333 0.82 PDE4A (0.46) ADORA2AADORA2BPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 87 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9725474-B2 Modified nucleic acid TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-08-08 US claimed
EP-1419247-A2 METHOD FOR THE PRODUCTION OF NUCLEIC ACIDS CONSISTING OF STOCHASTICALLY COMBINED PARTS OF SOURCE NUCLEIC ACIDS Direvo Biotech AG (DE) 2004-05-19 EP claimed
WO-2003012100-A2 METHOD FOR THE PRODUCTION OF NUCLEIC ACIDS CONSISTING OF STOCHASTICALLY COMBINED PARTS OF SOURCE NUCLEIC ACIDS DIREVO BIOTECH AG (DE) 2003-02-13 WO claimed
EP-4658753-A1 CHLORELLA MICROALGAE Algenuity BV (NL) 2025-12-10 EP disclosed
EP-4658093-A1 FOOD COMPOSITION COMPRISING CHLOROPHYLL-DEFICIENT CHLORELLA BIOMASS WITH HIGH PROTEIN CONTENT >50WT% Unilever IP Holdings B.V. (NL) 2025-12-10 EP disclosed
EP-4658084-A1 FOOD COMPOSITION Unilever IP Holdings B.V. (NL) 2025-12-10 EP disclosed
EP-4658754-A1 ALGAE BIOMASS Algenuity BV (NL) 2025-12-10 EP disclosed
WO-2025082420-A1 AQUEOUS EMULSION, METHOD FOR PREPARING THE SAME, COATING COMPOSITION AND ARTICLE GUANGDONG HUARUN PAINTS CO., LTD. (CN) 2025-04-24 WO disclosed
US-20250027033-A1 MODIFIED STRAINS OF CHLORELLA VULGARIS AND METHOD OF PRODUCTION ALGENUITY HOLDINGS LTD (GB) 2025-01-23 US disclosed
WO-2024160737-A1 FOOD COMPOSITION COMPRISING CHLOROPHYLL-DEFICIENT CHLORELLA BIOMASS WITH HIGH PROTEIN CONTENT >50WT% UNILEVER IP HOLDINGS B.V. (NL) 2024-08-08 WO disclosed
WO-2024160738-A1 FOOD COMPOSITION UNILEVER IP HOLDINGS B.V. (NL) 2024-08-08 WO disclosed
WO-2002004621-A2 METHODS OF CREATING CONSTRUCTS USEFUL FOR INTRODUCING SEQUENCES INTO EMBRYONIC STEM CELLS DELTAGEN, INC. (US) 2002-01-17 WO disclosed
WO-2001092308-A2 CYSTINE-KNOT POLYPEPTIDES: CLOAKED-2 MOLECULES AND USES THEREOF AMGEN, INC. (US) 2001-12-06 WO disclosed
US-6303618-B1 ADMINISTERING PURINE COMPOUND WHICH INHIBITS CYCLIC DEPENDENT KINASE ACTIVITY FOR THERAPY OF TUMOR OR OTHER CELL PROLIFERATION DISORDER CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2001-10-16 US disclosed
EP-1127165-A1 METHOD AND TEST KIT FOR ANALYZING DNS REPAIR Nehls, Peter (DE) 2001-08-29 EP disclosed
WO-2000026402-A1 METHOD AND TEST KIT FOR ANALYZING DNS REPAIR NEHLS PETER (DE) 2000-05-11 WO disclosed
WO-2000017220-A1 ANTISENSE MODULATION OF FAN EXPRESSION ISIS PHARMACEUTICALS, INC. (US) 2000-03-30 WO disclosed
WO-1999002162-A9 CYCLIN DEPENDENT KINASE INHIBITING PURINE DERIVATIVES CANCER RES CAMPAIGN TECH (GB) 1999-07-29 WO disclosed
EP-0846772-A1 Multifunctional ligand system for cell-specific transfer of nucleic acid HOECHST AKTIENGESELLSCHAFT (DE) 1998-06-10 EP disclosed
EP-0702683-A1 06-SUBSTITUTED GUANINE DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND THEIR USE IN TREATING TUMOUR CELLS CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 1996-03-27 EP disclosed