SCHEMBL5503704

SCHEMBL5503704

O=C1CC=CC2=C1CNc1cc(Cl)ccc1N2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 2/20 0.38
AHR P35869 2/20 0.36
CMA1 P23946 1/20 0.36
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
CES1 P23141 2/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
TGM2 P21980 1/20 0.33
LIMK1 P53667 1/20 0.32
GAA P10253 2/20 0.32
MAPT P10636 2/20 0.32
PDE7A Q13946 2/20 0.31
GABRP O00591 1/20 0.30
GABRD O14764 1/20 0.30
GABRA1 P14867 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7982185 0.82 MEN1 (0.48) AHRMEN1KMT2AMAPTMAPK13
SCHEMBL1290778 0.80 SMYD3 (0.36) MEN1KMT2A
SCHEMBL1290780 0.73 ITGB3 (0.31) MEN1KMT2AMAPT
SCHEMBL31332320 0.72 CA12 (0.36) AHRCMA1KMT2ACA12CA2
SCHEMBL1319879 0.72 AHR (0.55) CHEK1AHRCMA1MEN1KMT2A
SCHEMBL30509190 0.65 AHR (0.55) CHEK1AHRCMA1MEN1KMT2A
SCHEMBL11463464 0.65 AHR (0.55) CHEK1AHRCMA1MEN1KMT2A
SCHEMBL29532858 0.65 CHEK1 (0.49) CHEK1AHRCMA1MEN1KMT2A
SCHEMBL3522841 0.65 CHEK1 (0.49) CHEK1AHRCMA1MEN1KMT2A
SCHEMBL28552531 0.64 AHR (0.50) AHRMEN1KMT2ACES1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756070-A2 CRYSTALLINE FORMS OF N-DESMETHYLCLOZAPINE Acadia Pharmaceuticals Inc. (US) 2007-02-28 EP disclosed
WO-2006001866-A2 CRYSTALLINE FORMS OF N-DESMETHYLCLOZAPINE ACADIA PHARMACEUTICALS INC. (US) 2006-01-05 WO disclosed