SCHEMBL5504103

SCHEMBL5504103

CCCN1CCN(c2cccc(C(=O)C(F)(F)F)c2F)CC1.CCN1CCN(c2cccc(C(=O)C(F)(F)F)c2F)CC1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 9/20 0.45
DRD3 P35462 4/20 0.45
TTR P02766 1/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HTR1A P08908 3/20 0.41
DRD4 P21917 2/20 0.41
HTR2B P41595 1/20 0.41
ALDH1A1 P00352 1/20 0.40
HTR2A P28223 2/20 0.39
HTR6 P50406 1/20 0.39
HTR2C P28335 1/20 0.39
CHRM5 P08912 3/20 0.39
CHRM1 P11229 3/20 0.39
CHRM3 P20309 3/20 0.39
CHRM4 P08173 1/20 0.39
SIGMAR1 Q99720 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2782660 0.96 DRD2 (0.48) DRD2DRD3TTRHTR1ADRD4
SCHEMBL2782086 0.94 TTR (0.46) DRD2DRD3TTRNPC1RAB9A
SCHEMBL5519082 0.88 DRD2 (0.45) DRD2DRD3ALDH1A1HTR2AHTR6
SCHEMBL5501574 0.84 DRD2 (0.42) DRD2DRD3NPC1RAB9ASMN1; SMN2
SCHEMBL2783650 0.84 DRD2 (0.48) DRD2DRD3HTR1ADRD4ALDH1A1
SCHEMBL2782744 0.84 DRD2 (0.52) DRD2DRD3TTRHTR1ADRD4
SCHEMBL2784018 0.84 DRD2 (0.48) DRD2DRD3TTRHTR1ADRD4
SCHEMBL2784733 0.83 DRD2 (0.60) DRD2DRD3HTR1ADRD4HTR2B
SCHEMBL2781571 0.82 NPC1 (0.50) TTRNPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL2783413 0.82 ALDH1A1 (0.44) NPC1RAB9ASMN1; SMN2ALDH1A1CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773772-A1 NEW DISUBSTITUTED PHENYLPIPERIDINES/PIPERAZINES AS MODULATORS OF DOPAMINE NEUROTRANSMISSION A. CARLSSON RESEARCH AB (SE) 2007-04-18 EP claimed
WO-2005121087-A1 NEW DISUBSTITUTED PHENYLPIPERIDINES/PIPERAZINES AS MODULATORS OF DOPAMINE NEUROTRANSMISSION A. CARLSSON RESEARCH AB (SE) 2005-12-22 WO claimed