SCHEMBL5504183

SCHEMBL5504183

Cc1nc2ccccc2c2cn(-c3ccccc3)nc12

nearest known ligand 0.68

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 19/20 0.68
ADORA2A P29274 13/20 0.68
ADORA1 P30542 6/20 0.68
CNR1 P21554 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5505166 0.77 ADORA3 (0.62) ADORA3ADORA2AADORA1
SCHEMBL31060487 0.74 ADORA3 (1.00) ADORA3ADORA2AADORA1
SCHEMBL29602474 0.73 ADORA2A (0.51) ADORA3ADORA2AADORA1CNR1
SCHEMBL2974505 0.73 ADORA3 (0.49) ADORA3ADORA2AADORA1CNR1
SCHEMBL31061120 0.71 ADORA3 (1.00) ADORA3ADORA2AADORA1
SCHEMBL5505165 0.70 ADORA3 (0.47) ADORA3ADORA2AADORA1CNR1
SCHEMBL85621 0.68 GPR3 (1.00) ADORA3
SCHEMBL5503114 0.68 ADORA3 (1.00) ADORA3ADORA2AADORA1CNR1
SCHEMBL17335816 0.68 KDM4E (0.60) ADORA3ADORA1CNR1
SCHEMBL2979520 0.67 ESR2 (0.62) ADORA3ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863813-A2 PYRAZOLO[3,4-C]QUINOLINES, PYRAZOLO[3,4-C]NAPHTHYRIDINES, ANALOGS THEREOF, AND METHODS Coley Pharmaceutical Group, Inc. (US) 2007-12-12 EP disclosed
WO-2006107771-A2 PYRAZOLO[3,4-c]QUINOLINES, PYRAZOLO[3,4-c]NAPHTHYRIDINES, ANALOGS THEREOF, AND METHODS COLEY PHARMACEUTICAL GROUP, INC. (US) 2006-10-12 WO disclosed