SCHEMBL5503114

SCHEMBL5503114

Cn1c(=O)c2nn(-c3ccccc3)cc2c2ccccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 11/20 1.00
CA9 Q16790 1/20 0.49
ADORA1 P30542 4/20 0.48
ALDH1A1 P00352 2/20 0.48
KMT2A Q03164 1/20 0.48
ADORA2A P29274 3/20 0.48
PGR P06401 1/20 0.48
KDM4E B2RXH2 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
HPGD P15428 1/20 0.46
TSHR P16473 1/20 0.46
CYP2C19 P33261 1/20 0.46
HSD17B10 Q99714 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
CNR1 P21554 1/20 0.43
GPR3 P46089 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5508801 0.83 ADORA3 (0.83) ADORA3CA9ADORA1ALDH1A1ADORA2A
SCHEMBL5511769 0.82 ADORA3 (1.00) ADORA3CA9ADORA1ALDH1A1KMT2A
SCHEMBL5513775 0.80 ADORA3 (0.86) ADORA3ALDH1A1KMT2APGRKDM4E
Hydrochloric Acid SCHEMBL5507703 0.78 ADORA3 (0.71) ADORA3CA9ADORA1ADORA2APGR
SCHEMBL5503857 0.72 ADORA3 (0.64) ADORA3CA9ADORA1ADORA2AKDM4E
SCHEMBL31276757 0.69 GPR3 (0.65) ADORA3ALDH1A1KMT2APGRKDM4E
SCHEMBL346785 0.69 GPR3 (0.65) ADORA3ALDH1A1KMT2APGRKDM4E
SCHEMBL728937 0.69 ADORA3 (0.80) ADORA3ADORA1
SCHEMBL14802110 0.68 ADORA3 (0.55) ADORA3CA9ADORA1ADORA2AKDM4E
SCHEMBL5504183 0.68 ADORA3 (0.68) ADORA3ADORA1ADORA2ACNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863813-A2 PYRAZOLO[3,4-C]QUINOLINES, PYRAZOLO[3,4-C]NAPHTHYRIDINES, ANALOGS THEREOF, AND METHODS Coley Pharmaceutical Group, Inc. (US) 2007-12-12 EP disclosed
WO-2006107771-A2 PYRAZOLO[3,4-c]QUINOLINES, PYRAZOLO[3,4-c]NAPHTHYRIDINES, ANALOGS THEREOF, AND METHODS COLEY PHARMACEUTICAL GROUP, INC. (US) 2006-10-12 WO disclosed