SCHEMBL5504539

SCHEMBL5504539

O=CCc1cccc(-c2ccncc2)c1F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 1/20 0.36
KCNH2 Q12809 1/20 0.36
MAPK14 Q16539 3/20 0.36
PIK3CD O00329 1/20 0.35
PRKCI P41743 1/20 0.33
EGFR P00533 1/20 0.33
IDO1 P14902 1/20 0.33
PTPN5 P54829 4/20 0.32
RAB9A P51151 3/20 0.32
NR4A2 P43354 1/20 0.32
ALDH1A1 P00352 2/20 0.32
NPC1 O15118 2/20 0.32
PKM P14618 1/20 0.32
KMT2A Q03164 1/20 0.32
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32
MAPK10 P53779 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HSD17B10 Q99714 1/20 0.32
GCGR P47871 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2041153 0.80 DPP4 (0.47) KCNA5KCNH2MAPK14PIK3CDPRKCI
SCHEMBL23175855 0.77 PRMT6 (0.35) KCNA5KCNH2PIK3CDPRKCIIDO1
SCHEMBL27190814 0.73 AKR1B1 (0.32)
SCHEMBL1807270 0.71 CES2 (0.39) IDO1ALDH1A1SMN1; SMN2
SCHEMBL3637569 0.71 NPC1 (0.46) MAPK14PIK3CDRAB9ANPC1PKM
SCHEMBL3904012 0.71 CYP46A1 (0.36) MAPK14IDO1ALDH1A1KMT2AMAPT
SCHEMBL27893591 0.71 ROCK1 (0.41) ALDH1A1KMT2AMAPTSMN1; SMN2HSD17B10
SCHEMBL27893610 0.71 GPBAR1 (0.38) KCNA5KCNH2MAPK14PTPN5
SCHEMBL2039805 0.71 ROCK2 (0.41) MAPK14PRKCIKMT2AHSD17B10
SCHEMBL1980395 0.70 CES2 (0.38) IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773772-A1 NEW DISUBSTITUTED PHENYLPIPERIDINES/PIPERAZINES AS MODULATORS OF DOPAMINE NEUROTRANSMISSION A. CARLSSON RESEARCH AB (SE) 2007-04-18 EP disclosed
WO-2005121087-A1 NEW DISUBSTITUTED PHENYLPIPERIDINES/PIPERAZINES AS MODULATORS OF DOPAMINE NEUROTRANSMISSION A. CARLSSON RESEARCH AB (SE) 2005-12-22 WO disclosed