SCHEMBL5504641

SCHEMBL5504641

CCOc1c(C(N)=O)cccc1-c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.57
ALDH1A1 P00352 2/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
CYP3A4 P08684 2/20 0.45
KDM4E B2RXH2 2/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2D6 P10635 2/20 0.45
CYP2C9 P11712 2/20 0.45
CYP2C19 P33261 2/20 0.45
TDP1 Q9NUW8 2/20 0.45
HPGD P15428 1/20 0.45
LMNA P02545 2/20 0.44
LTB4R2 Q9NPC1 1/20 0.43
HNF4A P41235 1/20 0.42
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
NR1I2 O75469 1/20 0.42
CHRM2 P08172 1/20 0.42
ADRA2A P08913 1/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5156328 0.88 HNF4A (0.53) BCAT2ALDH1A1L3MBTL1CYP3A4KDM4E
SCHEMBL30013864 0.87 SLC6A3 (0.48) BCAT2ALDH1A1L3MBTL1CYP3A4CYP1A2
SCHEMBL1667777 0.84 BCAT2 (0.56) BCAT2KDM4EPARP1
SCHEMBL30504310 0.83 BCAT2 (0.62) BCAT2ALDH1A1L3MBTL1KDM4EHNF4A
SCHEMBL3975515 0.82 BCAT2 (0.54) BCAT2L3MBTL1CYP3A4KDM4ETDP1
SCHEMBL3973836 0.82 BCAT2 (0.54) BCAT2ALDH1A1L3MBTL1KDM4ETDP1
Hydrochloric Acid SCHEMBL30628503 0.81 BCAT2 (0.61) BCAT2ALDH1A1L3MBTL1KDM4EHNF4A
Hydrochloric Acid SCHEMBL30504328 0.81 BCAT2 (0.61) BCAT2ALDH1A1L3MBTL1KDM4EHNF4A
SCHEMBL13828076 0.80 ALDH1A1 (0.46) ALDH1A1L3MBTL1CYP3A4KDM4ECYP1A2
SCHEMBL22468856 0.79 PARP10 (0.53) BCAT2ALDH1A1LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1814866-A2 GONADOTROPIN RELEASING HORMONE RECEPTOR ANTAGONISTS Wyeth a Corporation of the State of Delaware (US) 2007-08-08 EP claimed
WO-2006058012-A2 GONADOTROPIN RELEASING HORMONE RECEPTOR ANTAGONISTS WYETH (US) 2006-06-01 WO claimed
WO-2004039795-A2 AMIDE COMPOUNDS FOR THE TREATMENT OF HYPERLIPIDEMIA FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-05-13 WO disclosed