SCHEMBL5504740

SCHEMBL5504740

NC(=O)CCNCCc1ccc(F)cc1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.54
ALDH1A1 P00352 1/20 0.54
HPGD P15428 1/20 0.51
CA12 O43570 2/20 0.49
CA1 P00915 2/20 0.49
CA2 P00918 2/20 0.49
CA4 P22748 1/20 0.49
PLAAT3 P53816 1/20 0.48
PLAAT5 Q96KN8 1/20 0.48
PLAAT2 Q9NWW9 1/20 0.48
PLAAT4 Q9UL19 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.47
TAAR1 Q96RJ0 1/20 0.47
KMT2A Q03164 1/20 0.45
CA9 Q16790 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4462532 0.84 KDM4E (0.55) KDM4EALDH1A1HPGDCA12CA1
SCHEMBL3824789 0.82 SIGMAR1 (0.55) KDM4EALDH1A1CA12CA1CA2
SCHEMBL2466699 0.81 FFAR1 (0.55) ALDH1A1HPGDPLAAT3PLAAT5PLAAT2
SCHEMBL658360 0.80 LMNA (0.54) HPGDTAAR1
SCHEMBL31103545 0.79 HPGD (0.68) HPGDCA12CA1CA2PLAAT3
SCHEMBL1478337 0.78 NAAA (0.51) HPGDTAAR1
SCHEMBL29655674 0.77 NAAA (0.50) TAAR1
SCHEMBL14893159 0.77 HPGD (0.60) ALDH1A1HPGDCA12CA1CA2
SCHEMBL31577212 0.77 NAAA (0.50) TAAR1
SCHEMBL29655601 0.77 NAAA (0.50) TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1799645-A2 PROCESSES AND INTERMEDIATES FOR PREPARING CYSTEINE PROTEASE INHIBITORS Bayer Schering Pharma Aktiengesellschaft (DE) 2007-06-27 EP disclosed
WO-2006034004-A2 PROCESSES AND INTERMEDIATES FOR PREPARING CYSTEINE PROTEASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 2006-03-30 WO disclosed