SCHEMBL5505886

SCHEMBL5505886

O=C(CCC(=O)c1ccc(F)cc1)c1ccccc1.O=C(CCC(=O)c1ccc(N2CCCCC2)cc1)c1ccccc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.69
NPC1 O15118 5/20 0.66
RAB9A P51151 5/20 0.66
ALDH1A1 P00352 5/20 0.63
TP53 P04637 4/20 0.63
MAPT P10636 3/20 0.63
HPGD P15428 2/20 0.63
TSHR P16473 2/20 0.63
MAPK1 P28482 2/20 0.63
KDM4E B2RXH2 1/20 0.63
CASP1 P29466 1/20 0.63
CASP7 P55210 1/20 0.63
NPSR1 Q6W5P4 1/20 0.63
SMN1; SMN2 Q16637 3/20 0.60
ALOX15 P16050 2/20 0.60
LMNA P02545 1/20 0.60
STAT1 P42224 1/20 0.60
HSD17B10 Q99714 1/20 0.60
L3MBTL1 Q9Y468 1/20 0.60
POLB P06746 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4472849 0.93 ALDH1A1 (0.70) HTR1ANPC1RAB9AALDH1A1TP53
SCHEMBL4485908 0.81 RAB9A (0.69) HTR1ANPC1RAB9AALDH1A1MAPT
SCHEMBL3090713 0.81 POLB (0.77) HTR1ANPC1RAB9AALDH1A1MAPT
SCHEMBL4038422 0.80 NPC1 (1.00) NPC1RAB9AALDH1A1TP53MAPT
SCHEMBL14982135 0.78 NPC1 (0.77) NPC1RAB9AALDH1A1TP53MAPT
SCHEMBL2742812 0.78 NPC1 (0.96) NPC1RAB9AALDH1A1TP53MAPT
SCHEMBL11832194 0.78 HTR1A (0.65) HTR1AALDH1A1MAPTHPGDTSHR
SCHEMBL10605457 0.77 RAB9A (0.61) NPC1RAB9AALDH1A1TP53MAPT
SCHEMBL11763488 0.77 RAB9A (0.61) NPC1RAB9AALDH1A1TP53MAPT
SCHEMBL4432092 0.77 HDAC1 (0.63) HTR1ANPC1RAB9AALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1848692-A1 AZOLYLACYLGUANIDINES AS ß-SECRETASE INHIBITORS Wyeth (US) 2007-10-31 EP disclosed
WO-2006088711-A1 AZOLYLACYLGUANIDINES AS β-SECRETASE INHIBITORS WYETH (US) 2006-08-24 WO disclosed