SCHEMBL5508917

SCHEMBL5508917

O=C(O)c1c(Cl)cc(F)c(F)c1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA4 P22748 2/20 0.40
DPP4 P27487 1/20 0.39
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
CES2 O00748 3/20 0.38
CES1 P23141 3/20 0.38
MEN1 O00255 1/20 0.36
CRHBP P24387 1/20 0.36
KMT2A Q03164 1/20 0.36
CRHR2 Q13324 1/20 0.36
KMO O15229 1/20 0.36
TTR P02766 1/20 0.35
TSHR P16473 1/20 0.34
ALDH1A1 P00352 3/20 0.34
KDM4E B2RXH2 1/20 0.34
HSD17B10 Q99714 1/20 0.34
MAPK1 P28482 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364018 0.79 CA1 (0.50) CA1CA2CA4KEAP1NFE2L2
SCHEMBL6725463 0.79 DPP4 (0.33) CA1CA2CA4DPP4KEAP1
SCHEMBL28205230 0.77 DPP4 (0.38) CA1CA2CA4DPP4KEAP1
SCHEMBL8377346 0.77 DPP4 (0.44) CA1CA2CA4DPP4KEAP1
SCHEMBL2926338 0.76 NOTUM (0.38) DPP4KMO
SCHEMBL26162974 0.76 CYP3A4 (0.42) CA1CA2CA4DPP4CES2
SCHEMBL5336692 0.76 KEAP1 (0.44) CA1CA2CA4KEAP1NFE2L2
SCHEMBL31041213 0.76 KEAP1 (0.44) CA1CA2CA4KEAP1NFE2L2
SCHEMBL6728940 0.75 AKR1C2 (0.37) DPP4KEAP1NFE2L2KMOALDH1A1
SCHEMBL5784974 0.75 DPP4 (0.43) DPP4KEAP1NFE2L2CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1114812-B1 PROCESSES FOR THE PREPARATION OF FLUORINATED BENZOIC ACIDS OTSUKA PHARMA CO LTD (JP) 2007-06-20 EP disclosed
US-6333431-B1 ALKYLATING TETRAFLUOROBENZOIC ACID OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2001-12-25 US disclosed
EP-1114812-A1 PROCESSES FOR THE PREPARATION OF FLUORINATED BENZOIC ACIDS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2001-07-11 EP disclosed