SCHEMBL5511036

SCHEMBL5511036

Cc1cc(NC(=O)C(C)(C)N)ccc1N1C(=S)CCC1C

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPY2R P49146 2/20 0.37
PDK1 Q15118 1/20 0.36
PDK2 Q15119 1/20 0.36
PDK3 Q15120 1/20 0.36
PDK4 Q16654 1/20 0.36
F10 P00742 3/20 0.35
HRH3 Q9Y5N1 6/20 0.35
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.33
RAB9A P51151 3/20 0.33
NPC1 O15118 2/20 0.33
AKR1C3 P42330 1/20 0.33
WDR5 P61964 1/20 0.33
ALDH1A1 P00352 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4479045 0.81 AR (0.52) F10MAPTRAB9ANPC1ALDH1A1
SCHEMBL5511183 0.76 NPC1 (0.41) NPY2RF10MAPTRAB9ANPC1
SCHEMBL5505029 0.73 WDR5 (0.41) NPY2RF10HRH3RAB9ANPC1
SCHEMBL5514263 0.72 F10 (0.53) NPY2RF10
SCHEMBL5568419 0.70 NPY2R (0.42) NPY2RF10MAPTRAB9ANPC1
SCHEMBL5565439 0.69 F10 (0.59) F10HRH3MAPTRAB9ANPC1
SCHEMBL5562241 0.69 NPY2R (0.41) NPY2RF10MAPTRAB9ANPC1
SCHEMBL5506905 0.67 F10 (0.46) NPY2RF10MAPTWDR5
SCHEMBL5510391 0.67 F10 (0.46) NPY2RF10WDR5
SCHEMBL849082 0.67 ALDH1A1 (0.54) MAPTRAB9ANPC1ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1747217-A1 NOVEL SUBSTITUTED THIOPHENECARBOXAMIDES, THEIR PRODUCTION AND THEIR USE AS MEDICAMENTS Boehringer Ingelheim International GmbH (DE) 2007-01-31 EP disclosed
WO-2005111029-A1 NOVEL SUBSTITUTED THIOPHENECARBOXAMIDES, THEIR PRODUCTION AND THEIR USE AS MEDICAMENTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-11-24 WO disclosed