SCHEMBL5511272

SCHEMBL5511272

CC(=O)NCCOC(=O)CC(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 4/20 0.43
MTNR1B P49286 4/20 0.43
MAPK1 P28482 2/20 0.40
TSHR P16473 2/20 0.40
USP2 O75604 1/20 0.40
ALOX15 P16050 1/20 0.40
HSD17B10 Q99714 1/20 0.40
KDM4E B2RXH2 1/20 0.40
HIF1A Q16665 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
ALDH1A1 P00352 3/20 0.38
TDP1 Q9NUW8 1/20 0.38
MMP1 P03956 1/20 0.36
MMP2 P08253 1/20 0.36
MMP3 P08254 1/20 0.36
MMP9 P14780 1/20 0.36
MMP13 P45452 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14679295 0.85 CYP2D6 (0.43) L3MBTL1ALDH1A1TDP1MMP1MMP2
SCHEMBL9853199 0.81 MTNR1A (0.50) MTNR1AMTNR1BMAPK1TSHRUSP2
SCHEMBL12341335 0.80 EPHX1 (0.49) TSHR
SCHEMBL20749852 0.80 MMP1 (0.38) KDM4EL3MBTL1ALDH1A1TDP1MMP1
Hydrochloric Acid SCHEMBL30512137 0.80 CACNA2D1 (0.46) MTNR1AMTNR1BMAPK1TSHRUSP2
SCHEMBL26478811 0.79 ZDHHC20 (0.42) MAPK1TSHRALDH1A1TDP1MMP1
SCHEMBL18378814 0.79 MMP1 (0.46) ALDH1A1TDP1MMP1MMP2MMP3
SCHEMBL22340363 0.78 MMP1 (0.37) KDM4EALDH1A1TDP1MMP1MMP2
SCHEMBL20954435 0.78 MTNR1A (0.47) MTNR1AMTNR1BMAPK1TSHRUSP2
SCHEMBL12523122 0.78 MAPK1 (0.44) MTNR1AMTNR1BMAPK1TSHRUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8367666-B2 3-carbamoyl-2-pyridone derivatives SHIONOGI & CO., LTD. (JP) 2013-02-05 US disclosed
US-8178681-B2 methyl 3-methyl-2-{[2-oxo-1-(2-oxo-ethyl)-1,2,5,6,7,8,9,10-octahydro-cycloocta[b]pyridine-3-carbonyl]-amino}-butyrate; cannabinoid receptor agonist; antiinflammatory agent, immunostimulant, analgesic; atopic dermatitis; excellent in photostability, and have excellent transdermal and oral absorbency SHIONOGI & CO., LTD. (JP) 2012-05-15 US disclosed