SCHEMBL5515933

SCHEMBL5515933

CNc1ccc(N)cc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCI P41743 1/20 0.37
ALDH1A1 P00352 5/20 0.37
MAPT P10636 5/20 0.37
MAPK1 P28482 3/20 0.37
TDP1 Q9NUW8 2/20 0.37
LMNA P02545 2/20 0.37
GFER P55789 1/20 0.37
ADRA2B P18089 1/20 0.36
APP P05067 2/20 0.36
CASP1 P29466 1/20 0.34
GAA P10253 4/20 0.34
ALOX15 P16050 2/20 0.34
HTT P42858 2/20 0.34
MAPK14 Q16539 1/20 0.34
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA9 Q16790 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5508382 0.82 ALDH1A1 (0.36) PRKCIALDH1A1MAPTMAPK1ADRA2B
SCHEMBL1662774 0.81 MAPK14 (0.41) ALDH1A1MAPTMAPK1TDP1LMNA
SCHEMBL8033091 0.78 PRKCI (0.41) PRKCIALDH1A1MAPTMAPK1TDP1
SCHEMBL12367898 0.77 ALDH1A1 (0.37) ALDH1A1MAPTMAPK1TDP1LMNA
SCHEMBL13718688 0.77 GSK3B (0.40) ALDH1A1MAPTMAPK1TDP1LMNA
SCHEMBL15384343 0.77 MAPT (0.42) ALDH1A1MAPTMAPK1TDP1LMNA
SCHEMBL239073 0.77 IDO1 (0.35) ALDH1A1MAPTMAPK1TDP1LMNA
SCHEMBL18403936 0.77 ADRA2B (0.37) ALDH1A1MAPTMAPK1TDP1LMNA
SCHEMBL784058 0.76 PRKCI (0.53) PRKCIALDH1A1MAPTMAPK1TDP1
SCHEMBL306848 0.76 HTT (0.50) ALDH1A1MAPTTDP1GAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3882245-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2021-09-22 EP disclosed
WO-2018089373-A9 STEROIDS AND PROTEIN-CONJUGATES THEREOF REGENERON PHARMACEUTICALS, INC. (US) 2018-07-12 WO disclosed
EP-3327016-A1 PREPARATION OF MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2018-05-30 EP disclosed
WO-2018089373-A2 STEROIDS AND PROTEIN-CONJUGATES THEREOF REGENERON PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed
US-7208559-B2 Ethylened polymer and molded object obtained therefrom MITSUI CHEMICALS, INC. (JP) 2007-04-24 US disclosed
US-20060135712-A1 Ethylened polymer and molded object obtained therefrom MITSUI CHEMICALS, INC. (JP) 2006-06-22 US disclosed