SCHEMBL5518909

SCHEMBL5518909

CC(C)c1nc(CC(=O)O)c(C(=O)O)s1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.34
AKR1B1 P15121 5/20 0.33
ALDH1A1 P00352 2/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
GABRR1 P24046 1/20 0.32
NPC1 O15118 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
NFKB1 P19838 1/20 0.31
RAB9A P51151 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31
POLB P06746 1/20 0.31
PTGDR2 Q9Y5Y4 3/20 0.31
TARBP2 Q15633 1/20 0.31
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9642950 0.84 PKM (0.35) PKMALDH1A1HPGDTSHRNPC1
SCHEMBL9644275 0.83 PKM (0.34) PKMALDH1A1HPGDTSHRTARBP2
SCHEMBL9644034 0.83 ALDH1A1 (0.37) PKMALDH1A1HPGDTSHRNPC1
SCHEMBL9644938 0.81 PKM (0.33) PKMALDH1A1HPGDTSHRNPC1
SCHEMBL5517320 0.81 GABRR1 (0.36) AKR1B1ALDH1A1GABRR1NPC1GAA
SCHEMBL9644069 0.80 SMN1; SMN2 (0.34) PKMALDH1A1HPGDTSHRNPC1
SCHEMBL5521343 0.79 GCK (0.36) AKR1B1ALDH1A1GABRR1NPC1GAA
SCHEMBL5517237 0.79 PTGDR2 (0.36) AKR1B1ALDH1A1GABRR1MAPTPOLB
SCHEMBL9644916 0.79 GABRP (0.40) PKMALDH1A1TSHRNPC1MAPT
SCHEMBL14215474 0.77 ALDH1A1 (0.40) PKMALDH1A1HPGDTSHRGABRR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8367666-B2 3-carbamoyl-2-pyridone derivatives SHIONOGI & CO., LTD. (JP) 2013-02-05 US disclosed
US-8367666-B2 3-carbamoyl-2-pyridone derivatives SHIONOGI & CO., LTD. (JP) 2013-02-05 US disclosed
US-8178681-B2 methyl 3-methyl-2-{[2-oxo-1-(2-oxo-ethyl)-1,2,5,6,7,8,9,10-octahydro-cycloocta[b]pyridine-3-carbonyl]-amino}-butyrate; cannabinoid receptor agonist; antiinflammatory agent, immunostimulant, analgesic; atopic dermatitis; excellent in photostability, and have excellent transdermal and oral absorbency SHIONOGI & CO., LTD. (JP) 2012-05-15 US disclosed
US-8178681-B2 methyl 3-methyl-2-{[2-oxo-1-(2-oxo-ethyl)-1,2,5,6,7,8,9,10-octahydro-cycloocta[b]pyridine-3-carbonyl]-amino}-butyrate; cannabinoid receptor agonist; antiinflammatory agent, immunostimulant, analgesic; atopic dermatitis; excellent in photostability, and have excellent transdermal and oral absorbency SHIONOGI & CO., LTD. (JP) 2012-05-15 US disclosed