SCHEMBL5525530

SCHEMBL5525530

NS(=O)(=O)c1cccc(-c2cccn2C(=O)O)c1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA2 P00918 13/20 0.46
CA1 P00915 12/20 0.46
CA9 Q16790 10/20 0.44
CA13 Q8N1Q1 3/20 0.44
IKBKB O14920 1/20 0.44
BRD4 O60885 1/20 0.43
CA12 O43570 7/20 0.42
MAPT P10636 1/20 0.42
CA4 P22748 3/20 0.41
CA14 Q9ULX7 2/20 0.41
CA7 P43166 2/20 0.39
CA3 P07451 1/20 0.39
CA6 P23280 1/20 0.39
CA5A P35218 1/20 0.39
PLA2G7 Q13093 1/20 0.39
CA5B Q9Y2D0 1/20 0.39
TTK P33981 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2916486 0.80 HSP90AA1 (0.48) CA2CA1CA9IKBKBBRD4
SCHEMBL31460477 0.79 PCSK9 (0.41)
SCHEMBL20557308 0.78 MAOA (0.46) CA2CA1CA9BRD4CA12
SCHEMBL30668584 0.75 PCSK9 (0.46) MAPT
SCHEMBL1926937 0.71 CA2 (0.67) CA2CA1CA9CA13IKBKB
SCHEMBL28032548 0.71 CA2 (0.73) CA2CA1CA9CA13CA12
SCHEMBL2942959 0.71 TP53 (0.47) MAPT
SCHEMBL1870487 0.69 CA2 (0.69) CA2CA1CA9CA12CA14
SCHEMBL15380745 0.69 PARP1 (0.46) MAPT
SCHEMBL4733938 0.67 CA2 (0.64) CA2CA1CA9CA13IKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1856096-A2 PHENYLGLYCINAMIDE DERIVATIVES USEFUL AS ANTICOAGULANTS Bristol-Myers Squibb Company (US) 2007-11-21 EP disclosed
WO-2006076246-A2 PHENYLGLYCINAMIDE DERIVATIVES USEFUL AS ANTICOAGULANTS BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-20 WO disclosed